Thapsigargin at Non-Cytotoxic Levels Induces a Potent Host Antiviral Response that Blocks Influenza A Virus Replication.


Journal

Viruses
ISSN: 1999-4915
Titre abrégé: Viruses
Pays: Switzerland
ID NLM: 101509722

Informations de publication

Date de publication:
27 09 2020
Historique:
received: 01 09 2020
revised: 21 09 2020
accepted: 24 09 2020
entrez: 30 9 2020
pubmed: 1 10 2020
medline: 17 2 2021
Statut: epublish

Résumé

Influenza A virus is a major global pathogen of humans, and there is an unmet need for effective antivirals. Current antivirals against influenza A virus directly target the virus and are vulnerable to mutational resistance. Harnessing an effective host antiviral response is an attractive alternative. We show that brief exposure to low, non-toxic doses of thapsigargin (TG), an inhibitor of the sarcoplasmic/endoplasmic reticulum (ER) Ca

Identifiants

pubmed: 32992478
pii: v12101093
doi: 10.3390/v12101093
pmc: PMC7600819
pii:
doi:

Substances chimiques

Antiviral Agents 0
Interferon Type I 0
Thapsigargin 67526-95-8
Interferons 9008-11-1
Sarcoplasmic Reticulum Calcium-Transporting ATPases EC 3.6.3.8
Interferon Lambda 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Medical Research Council
ID : MC_PC_18058
Pays : United Kingdom
Organisme : Biotechnology and Biological Sciences Research Council
ID : BB/L015293/1
Pays : United Kingdom

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Auteurs

Leah V Goulding (LV)

School of Veterinary Medicine and Science, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

Jiayun Yang (J)

School of Veterinary Medicine and Science, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

Zhimin Jiang (Z)

Key Laboratory of Animal Epidemiology, Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, No. 2 Yuanmingyuan West Road, Beijing 100193, China.

Hongyu Zhang (H)

Key Laboratory of Animal Epidemiology, Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, No. 2 Yuanmingyuan West Road, Beijing 100193, China.

Daniel Lea (D)

Advanced Data Analysis Centre, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

Richard D Emes (RD)

School of Veterinary Medicine and Science, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.
Advanced Data Analysis Centre, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

Tania Dottorini (T)

School of Veterinary Medicine and Science, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

Juan Pu (J)

Key Laboratory of Animal Epidemiology, Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, No. 2 Yuanmingyuan West Road, Beijing 100193, China.

Jinhua Liu (J)

Key Laboratory of Animal Epidemiology, Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, No. 2 Yuanmingyuan West Road, Beijing 100193, China.

Kin-Chow Chang (KC)

School of Veterinary Medicine and Science, University of Nottingham, Sutton Bonington Campus, Sutton Bonington LE12 5RD, UK.

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Classifications MeSH