Drug-induced cholestasis assay in primary hepatocytes.
Drug candidate selection
Drug safety evaluation
Drug-induced cholestasis
Drug-induced liver injury
In vitro toxicity
Primary hepatocytes
Journal
MethodsX
ISSN: 2215-0161
Titre abrégé: MethodsX
Pays: Netherlands
ID NLM: 101639829
Informations de publication
Date de publication:
2020
2020
Historique:
received:
15
07
2020
accepted:
23
09
2020
entrez:
22
10
2020
pubmed:
23
10
2020
medline:
23
10
2020
Statut:
epublish
Résumé
Drug-induced cholestasis (DIC) is a major cause of clinical failure of drug candidates. Numerous patients worldwide are affected when exposed to marketed drugs exhibiting a DIC signature. Prospective identification of DIC during early compound development remains challenging. Here we describe the optimized
Identifiants
pubmed: 33088729
doi: 10.1016/j.mex.2020.101080
pii: S2215-0161(20)30300-9
pmc: PMC7559231
doi:
Types de publication
Journal Article
Langues
eng
Pagination
101080Informations de copyright
© 2020 The Author(s). Published by Elsevier B.V.
Références
J Clin Pharmacol. 2006 Jun;46(6):628-34
pubmed: 16707409
J Antimicrob Chemother. 2009 Nov;64(5):1071-9
pubmed: 19710077
Am J Epidemiol. 2006 Apr 1;163(7):670-5
pubmed: 16410346
Drug Metab Dispos. 2016 Jan;44(1):16-27
pubmed: 26502773
Antimicrob Agents Chemother. 2003 May;47(5):1694-9
pubmed: 12709342
Toxicol Sci. 2010 Dec;118(2):485-500
pubmed: 20829430
JCI Insight. 2017 Mar 9;2(5):e90780
pubmed: 28289714
Drug Discov Today. 2012 May;17(9-10):475-85
pubmed: 22210121
Arch Toxicol. 2016 Dec;90(12):2979-3003
pubmed: 27659300
Pediatr Infect Dis J. 2016 Dec;35(12):1333-1335
pubmed: 27583590
Eur J Clin Pharmacol. 1999 Aug;55(6):461-7
pubmed: 10492060
Regul Toxicol Pharmacol. 2005 Aug;42(3):265-74
pubmed: 15979222
Drug Metab Dispos. 2016 Oct;44(10):1633-42
pubmed: 27417179
Crit Rev Toxicol. 2019 Jul;49(6):520-548
pubmed: 31589080
Curr Drug Metab. 2005 Apr;6(2):111-25
pubmed: 15853763
CPT Pharmacometrics Syst Pharmacol. 2014 Jul 09;3:e124
pubmed: 25006781
J Chromatogr B Analyt Technol Biomed Life Sci. 2013 Dec 30;942-943:53-62
pubmed: 24212143
J Pharm Sci. 2013 Sep;102(9):2953-94
pubmed: 23798314
Clin Pharmacol Ther. 2012 Jul;92(1):50-61
pubmed: 22644330
Clin Pharmacokinet. 1989 Apr;16(4):193-214
pubmed: 2656049
J Pharm Pharmacol. 1993 Sep;45(9):825-9
pubmed: 7903373
Methods Mol Biol. 2015;1250:363-76
pubmed: 26272158
Br J Clin Pharmacol. 1982 May;13(5):685-91
pubmed: 7082537
Clin Pharmacol Ther. 2006 Dec;80(6):657-67
pubmed: 17178266
Methods Mol Biol. 2010;640:1-40
pubmed: 20645044
Aliment Pharmacol Ther. 1998 Apr;12(4):373-6
pubmed: 9690728
Clin Pharmacokinet. 1998 Oct;35(4):275-91
pubmed: 9812178
Drug Metab Dispos. 2012 Jan;40(1):130-8
pubmed: 21965623
Sci Rep. 2016 Oct 19;6:35434
pubmed: 27759057
Handb Exp Pharmacol. 2010;(196):407-18
pubmed: 20020269
Toxicol Appl Pharmacol. 2014 Jan 1;274(1):124-36
pubmed: 24211272
BMC Bioinformatics. 2011 Mar 17;12:77
pubmed: 21414208
Toxicol In Vitro. 2016 Aug;34:179-186
pubmed: 27046439
J Pharmacol Toxicol Methods. 2015 May-Jun;73:63-71
pubmed: 25828992
Clin Chem Lab Med. 2003 Dec;41(12):1633-41
pubmed: 14708888
Expert Opin Drug Metab Toxicol. 2013 May;9(5):589-616
pubmed: 23452081
J Pharm Sci. 2013 Sep;102(9):3037-57
pubmed: 23653385
Appl Environ Microbiol. 1995 Apr;61(4):1614-9
pubmed: 7747975
J Chromatogr B Analyt Technol Biomed Life Sci. 2009 Nov 15;877(30):3920-5
pubmed: 19819765
Br J Pharmacol. 2008 Aug;154(7):1446-56
pubmed: 18587422
Clin Infect Dis. 2012 Nov;55(9):1270-2
pubmed: 22820540
World J Gastroenterol. 2009 Jul 7;15(25):3134-41
pubmed: 19575493
Toxicol In Vitro. 2004 Dec;18(6):869-77
pubmed: 15465654
Toxicol Sci. 2008 Sep;105(1):97-105
pubmed: 18524759
J Clin Psychopharmacol. 1989 Feb;9(1):4-8
pubmed: 2708554
N Engl J Med. 2006 Feb 16;354(7):731-9
pubmed: 16481640
Methods Mol Biol. 2015;1250:317-21
pubmed: 26272154
J Young Pharm. 2013 Mar;5(1):13-7
pubmed: 24023446
Methods Mol Biol. 2019;1981:335-350
pubmed: 31016665
J Chromatogr B Analyt Technol Biomed Life Sci. 2012 Jun 15;899:135-45
pubmed: 22664055
AIDS. 1999 Oct 22;13(15):2083-9
pubmed: 10546861
J Clin Pharmacol. 1997 Feb;37(2):108-15
pubmed: 9055136
J Chromatogr B Analyt Technol Biomed Life Sci. 2005 Nov 5;826(1-2):147-59
pubmed: 16182619
Best Pract Res Clin Haematol. 2004 Mar;17(1):139-52
pubmed: 15171963