The Adrenal Medulla Modulates Mechanical Allodynia in a Rat Model of Neuropathic Pain.


Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
06 Nov 2020
Historique:
received: 05 10 2020
revised: 31 10 2020
accepted: 04 11 2020
entrez: 11 11 2020
pubmed: 12 11 2020
medline: 18 3 2021
Statut: epublish

Résumé

We have investigated whether the stress response mediated by the adrenal medulla in rats subjected to chronic constriction injury of the sciatic nerve (CCI) modulates their nocifensive behavior. Treatment with SK29661 (300 mg/kg; intraperitoneal (I.P.)), a selective inhibitor of phenylethanolamine N-methyltransferase (PNMT) that converts noradrenaline (NA) into adrenaline (A), fully reverted mechanical allodynia in the injured hind paw without affecting mechanical sensitivity in the contralateral paw. The effect was fast and reversible and was associated with a decrease in the A to NA ratio (A/NA) in the adrenal gland and circulating blood, an A/NA that was elevated by CCI. 1,2,3,4-tetrahydroisoquinoline-7-sulfonamide (SKF29661) did not affect exocytosis evoked by Ca

Identifiants

pubmed: 33171955
pii: ijms21218325
doi: 10.3390/ijms21218325
pmc: PMC7664230
pii:
doi:

Substances chimiques

Catecholamines 0
Phenylethanolamine N-Methyltransferase EC 2.1.1.28
Norepinephrine X4W3ENH1CV
Epinephrine YKH834O4BH

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Universidad Complutense de Madrid
ID : PR75/18-21593
Organisme : Ministerio de Ciencia e Innovación
ID : BFU2011-26253, BFU2015-70067-REDC, SAF2016-78892

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Auteurs

Marina Arribas-Blázquez (M)

Department of Pharmacology and Toxicology, Veterinary Faculty and Instituto Universitario de Investigación en Neuroquímica, Universidad Complutense de Madrid, 28040 Madrid, Spain.
Instituto de Investigación Sanitaria San Carlos, 28040 Madrid, Spain.

Luis Alcides Olivos-Oré (LA)

Department of Pharmacology and Toxicology, Veterinary Faculty and Instituto Universitario de Investigación en Neuroquímica, Universidad Complutense de Madrid, 28040 Madrid, Spain.
Instituto de Investigación Sanitaria San Carlos, 28040 Madrid, Spain.

María Victoria Barahona (MV)

Department of Pharmacology and Toxicology, Veterinary Faculty and Instituto Universitario de Investigación en Neuroquímica, Universidad Complutense de Madrid, 28040 Madrid, Spain.
Instituto de Investigación Sanitaria San Carlos, 28040 Madrid, Spain.

Aneta Wojnicz (A)

Departamento de Farmacología, Instituto Teófilo Hernando, Facultad de Medicina, Universidad Autónoma de Madrid, 28029 Madrid, Spain.
Instituto de Investigación Sanitaria, Hospital Universitario de La Princesa, 28006 Madrid, Spain.

Ricardo De Pascual (R)

Departamento de Farmacología, Instituto Teófilo Hernando, Facultad de Medicina, Universidad Autónoma de Madrid, 28029 Madrid, Spain.
Instituto de Investigación Sanitaria, Hospital Universitario de La Princesa, 28006 Madrid, Spain.

Mercedes Sánchez de la Muela (M)

Department of Animal Medicine and Surgery, Veterinary Faculty, Universidad Complutense de Madrid, 20040 Madrid, Spain.

Antonio G García (AG)

Departamento de Farmacología, Instituto Teófilo Hernando, Facultad de Medicina, Universidad Autónoma de Madrid, 28029 Madrid, Spain.
Instituto de Investigación Sanitaria, Hospital Universitario de La Princesa, 28006 Madrid, Spain.

Antonio R Artalejo (AR)

Department of Pharmacology and Toxicology, Veterinary Faculty and Instituto Universitario de Investigación en Neuroquímica, Universidad Complutense de Madrid, 28040 Madrid, Spain.
Instituto de Investigación Sanitaria San Carlos, 28040 Madrid, Spain.

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Classifications MeSH