Kinetic Modelling and Test-Retest Reproducibility for the Dopamine D
Animals
Benzazepines
/ pharmacokinetics
Brain
/ diagnostic imaging
Carbon Radioisotopes
Disease Models, Animal
Gene Knock-In Techniques
Huntington Disease
/ diagnostic imaging
Male
Mice
Mice, Transgenic
Molecular Imaging
/ methods
Positron-Emission Tomography
/ methods
Receptors, Dopamine D1
/ antagonists & inhibitors
Reproducibility of Results
Tissue Distribution
D1R
Dopamine receptor
Huntington’s disease
Kinetic modelling
Mouse
Preclinical imaging
Q175DN
SCH23390
Test-retest
Journal
Molecular imaging and biology
ISSN: 1860-2002
Titre abrégé: Mol Imaging Biol
Pays: United States
ID NLM: 101125610
Informations de publication
Date de publication:
04 2021
04 2021
Historique:
received:
19
06
2020
accepted:
03
11
2020
revised:
29
10
2020
pubmed:
13
11
2020
medline:
16
11
2021
entrez:
12
11
2020
Statut:
ppublish
Résumé
Our aim in this study was to compare different non-invasive pharmacokinetic models and assess test-retest reproducibility of the radioligand [ Adult WT (n = 9) and HET (n = 14) mice underwent a 90-min [ For all models, we measured a significant decline in dopamine D Ninety-minute acquisition and the use of SRTM for pharmacokinetic modelling is recommended. [
Identifiants
pubmed: 33179158
doi: 10.1007/s11307-020-01561-1
pii: 10.1007/s11307-020-01561-1
pmc: PMC7910372
doi:
Substances chimiques
Benzazepines
0
Carbon Radioisotopes
0
Carbon-11
0
Receptors, Dopamine D1
0
SCH 23390
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
208-219Références
PLoS One. 2012;7(12):e49838
pubmed: 23284626
Mol Imaging Biol. 2020 Aug;22(4):854-863
pubmed: 31792838
J Nucl Med. 1998 May;39(5):792-7
pubmed: 9591577
Front Neural Circuits. 2013 Oct 11;7:152
pubmed: 24130517
Proc Natl Acad Sci U S A. 1993 Oct 1;90(19):8861-5
pubmed: 8415621
Mol Neurobiol. 2020 Apr;57(4):2038-2047
pubmed: 31912442
Eur J Pharmacol. 1992 Aug 14;219(1):45-52
pubmed: 1397049
J Huntingtons Dis. 2014;3(4):333-41
pubmed: 25575954
Eur J Nucl Med Mol Imaging. 2017 Jun;44(6):1025-1032
pubmed: 28197685
Psychopharmacology (Berl). 1993;113(2):149-56
pubmed: 7855175
Eur J Pharmacol. 1988 Jan 27;146(1):113-20
pubmed: 2895008
J Cereb Blood Flow Metab. 2001 Oct;21(10):1146-50
pubmed: 11598491
Biomed Res Int. 2013;2013:808713
pubmed: 24083242
J Cereb Blood Flow Metab. 2002 Dec;22(12):1440-52
pubmed: 12468889
J Neurochem. 1985 Nov;45(5):1601-11
pubmed: 2864398
J Neurosci. 2002 May 1;22(9):3708-19
pubmed: 11978847
Prog Brain Res. 2014;211:235-54
pubmed: 24968783
EJNMMI Res. 2018 Aug 2;8(1):74
pubmed: 30069645
Mol Imaging Biol. 2018 Feb;20(1):114-123
pubmed: 28631142
IEEE Trans Med Imaging. 2020 Jul;39(7):2518-2530
pubmed: 32070945
Curr Opin Investig Drugs. 2001 Nov;2(11):1582-91
pubmed: 11763161
Int J Rad Appl Instrum A. 1986;37(10):1039-43
pubmed: 3027000
PLoS One. 2012;7(12):e50717
pubmed: 23284644
J Cereb Blood Flow Metab. 2020 Jun;40(6):1351-1362
pubmed: 31307287
PLoS One. 2013 Jul 23;8(7):e69782
pubmed: 23936100
J Cereb Blood Flow Metab. 2003 Sep;23(9):1096-112
pubmed: 12973026
Neuropsychopharmacology. 1994 Dec;11(4):245-56
pubmed: 7531978
J Cereb Blood Flow Metab. 1996 Sep;16(5):834-40
pubmed: 8784228
Psychopharmacology (Berl). 2013 Jul;228(1):167-74
pubmed: 23460265
Neuroscientist. 2003 Oct;9(5):404-16
pubmed: 14580124
PLoS One. 2016 Feb 09;11(2):e0148839
pubmed: 26859386
Neurobiol Dis. 2010 Feb;37(2):356-61
pubmed: 19853661
Brain. 1997 Mar;120 ( Pt 3):503-14
pubmed: 9126061
Brain. 1999 Dec;122 ( Pt 12):2353-63
pubmed: 10581228
Neurosci Lett. 1988 Aug 31;91(2):142-7
pubmed: 2972942
Psychopharmacology (Berl). 1987;92(3):278-84
pubmed: 2957716
Brain. 1995 Jun;118 ( Pt 3):689-96
pubmed: 7600086
Ann Neurol. 1996 Jul;40(1):49-54
pubmed: 8687191
Neuroimage. 1997 Nov;6(4):279-87
pubmed: 9417971
J Nucl Med. 2016 May;57(5):792-8
pubmed: 26912432
Mol Imaging Biol. 2007 May-Jun;9(3):117-25
pubmed: 17473957
PLoS One. 2018 Oct 26;13(10):e0206613
pubmed: 30365550
Neuroscience. 2006 Apr 28;139(1):263-76
pubmed: 16310964
J Nucl Med. 1998 Dec;39(12):2061-8
pubmed: 9867142
PLoS One. 2018 Aug 17;13(8):e0200626
pubmed: 30118496
Pharmacol Ther. 2010 Oct;128(1):37-60
pubmed: 20547182
Mol Psychiatry. 2000 Nov;5(6):664-72
pubmed: 11126397
Neuroimage. 1996 Dec;4(3 Pt 1):153-8
pubmed: 9345505
J Neurophysiol. 2015 Apr 1;113(7):2953-66
pubmed: 25673747
J Pharmacol Exp Ther. 1992 Mar;260(3):1361-5
pubmed: 1347569
J Cereb Blood Flow Metab. 2010 May;30(5):985-93
pubmed: 20029452
J Nucl Med. 2017 Apr;58(4):617-622
pubmed: 27856625
J Cereb Blood Flow Metab. 2007 Oct;27(10):1733-41
pubmed: 17311076
Synapse. 1998 Sep;30(1):56-61
pubmed: 9704881
J Nucl Med. 2013 Jul;54(7):1127-34
pubmed: 23729696