Fragment-Based Identification of Ligands for Bromodomain-Containing Factor 3 of

BI-2536 Chagas disease Trypanosoma cruzi bromodomain-containing factor 3 fragment-based discovery

Journal

ACS infectious diseases
ISSN: 2373-8227
Titre abrégé: ACS Infect Dis
Pays: United States
ID NLM: 101654580

Informations de publication

Date de publication:
13 08 2021
Historique:
pubmed: 19 11 2020
medline: 10 9 2021
entrez: 18 11 2020
Statut: ppublish

Résumé

The

Identifiants

pubmed: 33203208
doi: 10.1021/acsinfecdis.0c00618
doi:

Substances chimiques

Ligands 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

2238-2249

Subventions

Organisme : Biotechnology and Biological Sciences Research Council
ID : BB/M015157/1
Pays : United Kingdom
Organisme : Cancer Research UK
Pays : United Kingdom

Auteurs

Corentine M C Laurin (CMC)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Joseph P Bluck (JP)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
Department of Biochemistry, University of Oxford, 3 Parks Road, Oxford OX1 3QU, UK.

Anthony K N Chan (AKN)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Michelle Keller (M)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Andrew Boczek (A)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Amy R Scorah (AR)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

K F Larissa See (KFL)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Laura E Jennings (LE)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

David S Hewings (DS)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Fern Woodhouse (F)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Jessica K Reynolds (JK)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Matthias Schiedel (M)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

Philip G Humphreys (PG)

GlaxoSmithKline R&D, Stevenage, Hertfordshire SG1 2NY, UK.

Philip C Biggin (PC)

Department of Biochemistry, University of Oxford, 3 Parks Road, Oxford OX1 3QU, UK.

Stuart J Conway (SJ)

Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.

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