Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors.
CCR2
CCR5 antagonists
PET
TAK-779
chemokine receptors
molecular imaging
radiolabeling
Journal
ChemMedChem
ISSN: 1860-7187
Titre abrégé: ChemMedChem
Pays: Germany
ID NLM: 101259013
Informations de publication
Date de publication:
17 02 2021
17 02 2021
Historique:
received:
16
09
2020
revised:
04
11
2020
pubmed:
19
11
2020
medline:
4
11
2021
entrez:
18
11
2020
Statut:
ppublish
Résumé
Herein we report the design and synthesis of a series of highly selective CCR2 antagonists as
Identifiants
pubmed: 33205603
doi: 10.1002/cmdc.202000728
pmc: PMC7983900
doi:
Substances chimiques
CCR2 protein, human
0
Radiopharmaceuticals
0
Receptors, CCR2
0
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
640-645Subventions
Organisme : Brazilian Doctoral Scholarship Program in Federal Republic of Germany
ID : 290265/2017-7
Organisme : NIDA NIH HHS
ID : HHSN271201800023C
Pays : United States
Informations de copyright
© 2020 The Authors. ChemMedChem published by Wiley-VCH GmbH.
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