Mechanisms of Resistance to Prostate-Specific Membrane Antigen-Targeted Radioligand Therapy in a Mouse Model of Prostate Cancer.

DNA damage response [177Lu]Lu-PSMA [225Ac]Ac-PSMA prostate cancer proteomics/phosphoproteomics

Journal

Journal of nuclear medicine : official publication, Society of Nuclear Medicine
ISSN: 1535-5667
Titre abrégé: J Nucl Med
Pays: United States
ID NLM: 0217410

Informations de publication

Date de publication:
01 07 2021
Historique:
received: 02 09 2020
revised: 11 11 2020
pubmed: 6 12 2020
medline: 6 1 2022
entrez: 5 12 2020
Statut: ppublish

Résumé

Prostate-specific membrane antigen (PSMA)-targeted radioligand therapy (RLT) is effective against prostate cancer (PCa), but all patients relapse eventually. Poor understanding of the underlying resistance mechanisms represents a key barrier to development of more effective RLT. We investigate the proteome and phosphoproteome in a mouse model of PCa to identify signaling adaptations triggered by PSMA RLT.

Identifiants

pubmed: 33277393
pii: jnumed.120.256263
doi: 10.2967/jnumed.120.256263
pmc: PMC8882874
doi:

Substances chimiques

Prostate-Specific Antigen EC 3.4.21.77

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

989-995

Subventions

Organisme : NCI NIH HHS
ID : P30 CA016042
Pays : United States
Organisme : NCI NIH HHS
ID : P50 CA211015
Pays : United States
Organisme : NCI NIH HHS
ID : P50 CA092131
Pays : United States

Informations de copyright

© 2021 by the Society of Nuclear Medicine and Molecular Imaging.

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Auteurs

Andreea D Stuparu (AD)

Atreca Inc., South San Francisco, California.

Joseph R Capri (JR)

AstraZeneca, Chemical Biology Group, Waltham, Massachusetts.

Catherine A L Meyer (CAL)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.

Thuc M Le (TM)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.

Susan L Evans-Axelsson (SL)

Department of Translational Medicine, Division of Urological Cancers, Skåne University Hospital Malmö, Lund University, Lund, Sweden.

Kyle Current (K)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.

Mark Lennox (M)

School of Electronics, Electrical Engineering, and Computer Science, Queen's University Belfast, Belfast, United Kingdom.

Christine E Mona (CE)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.
Department of Urology, Institute of Urologic Oncology, UCLA, Los Angeles, California; and.
Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, California.

Wolfgang P Fendler (WP)

Department of Nuclear Medicine, University of Duisburg-Essen and German Cancer Consortium-University Hospital Essen, Essen, Germany.

Jeremie Calais (J)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.
Department of Urology, Institute of Urologic Oncology, UCLA, Los Angeles, California; and.
Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, California.

Matthias Eiber (M)

Clinic for Nuclear Medicine, Technical University Munich, Munich, Germany.

Magnus Dahlbom (M)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.

Johannes Czernin (J)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.
Department of Urology, Institute of Urologic Oncology, UCLA, Los Angeles, California; and.
Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, California.

Caius G Radu (CG)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.
Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, California.

Katharina Lückerath (K)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California; klueckerath@mednet.ucla.edu.
Department of Urology, Institute of Urologic Oncology, UCLA, Los Angeles, California; and.
Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, California.

Roger Slavik (R)

Department of Molecular and Medical Pharmacology, David Geffen School of Medicine at UCLA, Los Angeles, California.

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Classifications MeSH