In vitro metabolism curcumin curcumin diethyl disuccinate liver S9 monoethylsuccinyl curcumin

Journal

Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923

Informations de publication

Date de publication:
2020
Historique:
received: 30 06 2020
accepted: 21 09 2020
entrez: 14 12 2020
pubmed: 15 12 2020
medline: 15 12 2020
Statut: epublish

Résumé

Liver S9 (LS9) is a nearly complete collection of all hepatic drug-metabolizing enzymes. It is a low-cost model for predicting drug metabolic activity. This study aimed to identify the suitability of using LS9 of different animal sources in drug metabolism profiling with respect to the possible translation of the

Identifiants

pubmed: 33312126
doi: 10.3389/fphar.2020.577998
pii: 577998
pmc: PMC7703437
doi:

Types de publication

Journal Article

Langues

eng

Pagination

577998

Informations de copyright

Copyright © 2020 Rojsitthisak, Jithavech, Ratnatilaka Na Bhuket, Supasena, Qiu, Ye, Wu and Wong.

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Auteurs

Ponsiree Jithavech (P)

Pharmaceutical Chemistry and Natural Products Program, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok, Thailand.
Natural Products for Ageing and Chronic Diseases Research Unit, Chulalongkorn University, Bangkok, Thailand.

Pahweenvaj Ratnatilaka Na Bhuket (P)

Natural Products for Ageing and Chronic Diseases Research Unit, Chulalongkorn University, Bangkok, Thailand.

Wiwat Supasena (W)

Natural Products for Ageing and Chronic Diseases Research Unit, Chulalongkorn University, Bangkok, Thailand.

Guanyinsheng Qiu (G)

College of Biological, Chemical Sciences and Engineering, Jiaxing University, Jiaxing, China.

Shengqing Ye (S)

School of Pharmaceutical and Materials Engineering & Institute for Advanced Studies, Taizhou University, Taizhou, China.

Jie Wu (J)

School of Pharmaceutical and Materials Engineering & Institute for Advanced Studies, Taizhou University, Taizhou, China.

Tin Wui Wong (TW)

Non-Destructive Biomedical and Pharmaceutical Research Centre, iPROMISE, Universiti Teknologi MARA, Puncak Alam, Malaysia.

Pornchai Rojsitthisak (P)

Natural Products for Ageing and Chronic Diseases Research Unit, Chulalongkorn University, Bangkok, Thailand.
Department of Food and Pharmaceutical Chemistry, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok, Thailand.

Classifications MeSH