Rationally designed N-phenylsulfonylindoles as a tool for the analysis of the non-basic 5-HT

Drug Design HEK293 Cells Humans Indoles / chemistry Ligands Molecular Dynamics Simulation Radioligand Assay Receptors, Serotonin / metabolism Structure-Activity Relationship

Journal

European journal of medicinal chemistry
ISSN: 1768-3254
Titre abrégé: Eur J Med Chem
Pays: France
ID NLM: 0420510

Informations de publication

Date de publication:
01 Jan 2021
Historique:
received: 30 04 2020
revised: 17 09 2020
accepted: 05 10 2020
entrez: 17 12 2020
pubmed: 18 12 2020
medline: 24 4 2021
Statut: ppublish

Résumé

Among all of the monoaminergic receptors, the 5-HT

Identifiants

DOI: 10.1016/j.ejmech.2020.112916 PMID: 33328102
pubmed: 33328102
pii: S0223-5234(20)30888-6
doi: 10.1016/j.ejmech.2020.112916
pii:
doi:

Substances chimiques

Indoles 0
Ligands 0
Receptors, Serotonin 0
serotonin 6 receptor 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

112916

Informations de copyright

Copyright © 2020 Elsevier Masson SAS. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of competing interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Jakub Staroń (J)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland. Electronic address: staron@if-pan.krakow.pl.

Ryszard Bugno (R)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Wojciech Pietruś (W)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Grzegorz Satała (G)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Stefan Mordalski (S)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Dawid Warszycki (D)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Agata Hogendorf (A)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Adam S Hogendorf (AS)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Justyna Kalinowska-Tłuścik (J)

Department of Crystal Chemistry and Crystal Physic Faculty of Chemistry, Jagiellonian University, Ingardena 3, 30-060, Kraków, Poland.

Tomasz Lenda (T)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

Bogusław Pilarski (B)

CERKO, 96/98 Zwycięstwa Avenue, 81-525, Gdynia, Poland.

Andrzej J Bojarski (AJ)

Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smętna Street, Poland.

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Classifications MeSH

questionsmedicales.fr › Techniques d'investigation › Développement de médicament › Découverte de médicament › Conception de médicament › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Cellules › Cellules épithéliales › Cellules HEK293 › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Primates › Haplorhini › Catarrhini › Hominidae › Humains › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Composés hétérocycliques › Composés hétérocycliques à cycles fusionnés › Composés hétérobicycliques › Indoles › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Ligands › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Sciences de l'information › Méthodologies informatiques › Simulation numérique › Simulation de dynamique moléculaire › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Techniques d'investigation › Techniques de laboratoire clinique › Dosage par compétition › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Protéines membranaires › Récepteurs de surface cellulaire › Récepteurs aux neuromédiateurs › Récepteurs sérotoninergiques › Rationally designed N-phenylsulfonylindoles as...
questionsmedicales.fr › Phénomènes physiologiques › Phénomènes pharmacologiques et toxicologiques › Phénomènes pharmacologiques › Relation structure-activité › Rationally designed N-phenylsulfonylindoles as...