Lithocholic Acid Derivatives as Potent Vitamin D Receptor Agonists.

Animals Crystallography, X-Ray Dose-Response Relationship, Drug HL-60 Cells Humans Ligands Lithocholic Acid / administration & dosage Molecular Structure Protein Binding Receptors, Calcitriol / agonists

Journal

Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531

Informations de publication

Date de publication:
14 01 2021
Historique:
pubmed: 29 12 2020
medline: 9 3 2021
entrez: 28 12 2020
Statut: ppublish

Résumé

Lithocholic acid (

Identifiants

DOI: 10.1021/acs.jmedchem.0c01420 PMID: 33369416
pubmed: 33369416
doi: 10.1021/acs.jmedchem.0c01420
doi:

Substances chimiques

Ligands 0
Receptors, Calcitriol 0
Lithocholic Acid 5QU0I8393U

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

516-526

Auteurs

Harue Sasaki (H)

Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Bunkyo, Tokyo 112-8610, Japan.

Hiroyuki Masuno (H)

Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University, 2-3-10 Kanda-Surugadai, Chiyoda-ku, Chiyoda, Tokyo 101-0062, Japan.

Haru Kawasaki (H)

Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Bunkyo, Tokyo 112-8610, Japan.

Ayana Yoshihara (A)

Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Bunkyo, Tokyo 112-8610, Japan.

Nobutaka Numoto (N)

Medical Research Institute, Tokyo Medical and Dental University, 1-5-45 Yushima, Bunkyo-ku, Bunkyo, Tokyo 113-8510, Japan.

Nobutoshi Ito (N)

Medical Research Institute, Tokyo Medical and Dental University, 1-5-45 Yushima, Bunkyo-ku, Bunkyo, Tokyo 113-8510, Japan.

Hiroaki Ishida (H)

Showa Pharmaceutical University, 3-3165 Higashi-Tamagawagakuen, Machidashi, Tokyo 194-8543, Japan.

Keiko Yamamoto (K)

Showa Pharmaceutical University, 3-3165 Higashi-Tamagawagakuen, Machidashi, Tokyo 194-8543, Japan.
ORCID: 0000-0001-6642-7961

Naoya Hirata (N)

Division of Pharmacology, National Institute of Health Sciences, 3-25-26 Tonomachi, Kawasaki-ku, Kawasaki, Kanagawa 210-9501, Japan.

Yasunari Kanda (Y)

Division of Pharmacology, National Institute of Health Sciences, 3-25-26 Tonomachi, Kawasaki-ku, Kawasaki, Kanagawa 210-9501, Japan.

Emiko Kawachi (E)

Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University, 2-3-10 Kanda-Surugadai, Chiyoda-ku, Chiyoda, Tokyo 101-0062, Japan.

Hiroyuki Kagechika (H)

Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University, 2-3-10 Kanda-Surugadai, Chiyoda-ku, Chiyoda, Tokyo 101-0062, Japan.
ORCID: 0000-0002-6747-1013

Aya Tanatani (A)

Department of Chemistry, Faculty of Science, Ochanomizu University, 2-1-1 Otsuka, Bunkyo-ku, Bunkyo, Tokyo 112-8610, Japan.
ORCID: 0000-0002-6667-8506

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Classifications MeSH

questionsmedicales.fr › Eucaryotes › Animaux › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Techniques d'investigation › Techniques de chimie analytique › Cristallographie aux rayons X › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Phénomènes physiologiques › Phénomènes pharmacologiques et toxicologiques › Phénomènes toxicologiques › Relation dose-effet des médicaments › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Cellules › Cellules myéloïdes › Cellules HL-60 › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Primates › Haplorhini › Catarrhini › Hominidae › Humains › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Ligands › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Composés polycycliques › Composés à cycles fusionnés › Stéroïdes › Cholanes › Acides choliques › Acide lithocholique › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Phénomènes chimiques › Structure moléculaire › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Métabolisme › Liaison aux protéines › Lithocholic Acid Derivatives as Potent Vitamin...
questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Récepteurs cytoplasmiques et nucléaires › Récepteur calcitriol › Lithocholic Acid Derivatives as Potent Vitamin...