Loss of POMC-mediated antinociception contributes to painful diabetic neuropathy.


Journal

Nature communications
ISSN: 2041-1723
Titre abrégé: Nat Commun
Pays: England
ID NLM: 101528555

Informations de publication

Date de publication:
18 01 2021
Historique:
received: 02 08 2019
accepted: 10 12 2020
entrez: 19 1 2021
pubmed: 20 1 2021
medline: 30 1 2021
Statut: epublish

Résumé

Painful neuropathy is a frequent complication in diabetes. Proopiomelanocortin (POMC) is an endogenous opioid precursor peptide, which plays a protective role against pain. Here, we report dysfunctional POMC-mediated antinociception in sensory neurons in diabetes. In streptozotocin-induced diabetic mice the Pomc promoter is repressed due to increased binding of NF-kB p50 subunit, leading to a loss in basal POMC level in peripheral nerves. Decreased POMC levels are also observed in peripheral nervous system tissue from diabetic patients. The antinociceptive pathway mediated by POMC is further impaired due to lysosomal degradation of μ-opioid receptor (MOR). Importantly, the neuropathic phenotype of the diabetic mice is rescued upon viral overexpression of POMC and MOR in the sensory ganglia. This study identifies an antinociceptive mechanism in the sensory ganglia that paves a way for a potential therapy for diabetic neuropathic pain.

Identifiants

pubmed: 33462216
doi: 10.1038/s41467-020-20677-0
pii: 10.1038/s41467-020-20677-0
pmc: PMC7814083
doi:

Substances chimiques

Oprm protein, mouse 0
Receptors, Opioid, mu 0
Streptozocin 5W494URQ81
Pro-Opiomelanocortin 66796-54-1

Types de publication

Journal Article Research Support, Non-U.S. Gov't Video-Audio Media

Langues

eng

Sous-ensembles de citation

IM

Pagination

426

Commentaires et corrections

Type : ErratumIn

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Auteurs

Divija Deshpande (D)

Department of Medicine I and Clinical Chemistry, University Hospital of Heidelberg, INF 410, Heidelberg, Germany.
Institute of Pharmacology, Heidelberg University, INF 366, Heidelberg, 69120, Germany.
Department of Microbiology, Infectious Diseases and Immunology, Charité -Universitätsmedizin Berlin, Hindenburgdamm 30, 12203, Berlin, Germany.

Nitin Agarwal (N)

Institute of Pharmacology, Heidelberg University, INF 366, Heidelberg, 69120, Germany.

Thomas Fleming (T)

Department of Medicine I and Clinical Chemistry, University Hospital of Heidelberg, INF 410, Heidelberg, Germany.
German Center for Diabetes Research (DZD), Neuherberg, Germany.

Claire Gaveriaux-Ruff (C)

Institut de Génétique et de Biologie Moléculaire et Cellulaire, Department of Translational Medicine and Neurogenetics, Illkirch, France.
Université de Strasbourg, Illkirch, France.
Centre National de la Recherche Scientifique, UMR7104, Illkirch, France.
Institut National de la Santé et de la Recherche Médicale, U1258, Illkirch, France.
Ecole Supérieure de Biotechnologie de Strasbourg, Illkirch, France.

Christoph S N Klose (CSN)

Department of Microbiology, Infectious Diseases and Immunology, Charité -Universitätsmedizin Berlin, Hindenburgdamm 30, 12203, Berlin, Germany.

Anke Tappe-Theodor (A)

Institute of Pharmacology, Heidelberg University, INF 366, Heidelberg, 69120, Germany.

Rohini Kuner (R)

Institute of Pharmacology, Heidelberg University, INF 366, Heidelberg, 69120, Germany.

Peter Nawroth (P)

Department of Medicine I and Clinical Chemistry, University Hospital of Heidelberg, INF 410, Heidelberg, Germany. peter.nawroth@med.uni-heidelberg.de.
German Center for Diabetes Research (DZD), Neuherberg, Germany. peter.nawroth@med.uni-heidelberg.de.
Joint Heidelberg-IDC Translational Diabetes Program, Helmholtz Zentrum, 85764, Neuherberg, Germany. peter.nawroth@med.uni-heidelberg.de.

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Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH