Radiosynthesis,
4R-tau
CBD-2115
PET
fluorine-18
tau
Journal
ACS chemical neuroscience
ISSN: 1948-7193
Titre abrégé: ACS Chem Neurosci
Pays: United States
ID NLM: 101525337
Informations de publication
Date de publication:
17 02 2021
17 02 2021
Historique:
pubmed:
27
1
2021
medline:
22
6
2021
entrez:
26
1
2021
Statut:
ppublish
Résumé
CBD-2115 was selected from a library of 148 compounds based on a pyridinyl-indole scaffold as a first-in-class 4R-tau radiotracer. In vitro binding assays showed [
Identifiants
pubmed: 33497190
doi: 10.1021/acschemneuro.0c00801
pmc: PMC9350900
mid: NIHMS1795861
doi:
Substances chimiques
Radiopharmaceuticals
0
tau Proteins
0
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
596-602Subventions
Organisme : NIA NIH HHS
ID : R01 AG052414
Pays : United States
Organisme : NIA NIH HHS
ID : R01 AG054473
Pays : United States
Organisme : NINDS NIH HHS
ID : U19 NS110456
Pays : United States
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