HPMA-Based Copolymers Carrying STAT3 Inhibitor Cucurbitacin-D as Stimulus-Sensitive Nanomedicines for Oncotherapy.

N-(2-hydroxypropyl) methacrylamide (HPMA) cucurbitacin-D immuno-oncotherapy pH-controlled release signal transducer and activator of transcription 3 (STAT3) inhibition

Journal

Pharmaceutics
ISSN: 1999-4923
Titre abrégé: Pharmaceutics
Pays: Switzerland
ID NLM: 101534003

Informations de publication

Date de publication:
28 Jan 2021
Historique:
received: 22 12 2020
revised: 22 01 2021
accepted: 23 01 2021
entrez: 2 2 2021
pubmed: 3 2 2021
medline: 3 2 2021
Statut: epublish

Résumé

The study describes the synthesis, physicochemical properties, and biological evaluation of polymer therapeutics based on

Identifiants

pubmed: 33525658
pii: pharmaceutics13020179
doi: 10.3390/pharmaceutics13020179
pmc: PMC7911143
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Grantová Agentura České Republiky
ID : 17-08084S
Organisme : Ministerstvo Školství, Mládeže a Tělovýchovy
ID : LTAUSA18083

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Auteurs

Marina R Tavares (MR)

Institute of Macromolecular Chemistry of the Czech Academy of Sciences, Heyrovského náměstí 2, CZ-162 06 Prague 6, Czech Republic.

Klára Hrabánková (K)

Institute of Microbiology of the Czech Academy of Sciences, Vídeňská 1083, CZ-142 20 Prague 4, Czech Republic.

Rafał Konefał (R)

Institute of Macromolecular Chemistry of the Czech Academy of Sciences, Heyrovského náměstí 2, CZ-162 06 Prague 6, Czech Republic.

Martin Kaňa (M)

Institute of Microbiology of the Czech Academy of Sciences, Vídeňská 1083, CZ-142 20 Prague 4, Czech Republic.

Blanka Říhová (B)

Institute of Microbiology of the Czech Academy of Sciences, Vídeňská 1083, CZ-142 20 Prague 4, Czech Republic.

Tomáš Etrych (T)

Institute of Macromolecular Chemistry of the Czech Academy of Sciences, Heyrovského náměstí 2, CZ-162 06 Prague 6, Czech Republic.

Milada Šírová (M)

Institute of Microbiology of the Czech Academy of Sciences, Vídeňská 1083, CZ-142 20 Prague 4, Czech Republic.

Petr Chytil (P)

Institute of Macromolecular Chemistry of the Czech Academy of Sciences, Heyrovského náměstí 2, CZ-162 06 Prague 6, Czech Republic.

Classifications MeSH