Simulation-Based Assessment of the Impact of Non-Adherence on Endoxifen Target Attainment in Different Tamoxifen Dosing Strategies.

model-informed precision dosing non-adherence pharmacokinetics pharmacometrics tamoxifen

Journal

Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453

Informations de publication

Date de publication:
03 Feb 2021
Historique:
received: 24 12 2020
revised: 22 01 2021
accepted: 29 01 2021
entrez: 6 2 2021
pubmed: 7 2 2021
medline: 7 2 2021
Statut: epublish

Résumé

Tamoxifen is widely used in breast cancer treatment and minimum steady-state concentrations of its active metabolite endoxifen (C

Identifiants

pubmed: 33546125
pii: ph14020115
doi: 10.3390/ph14020115
pmc: PMC7913149
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Freie Universität Berlin
ID : Open Access Fund

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Auteurs

Anna Mueller-Schoell (A)

Department of Clinical Pharmacy and Biochemistry, Institute of Pharmacy, Freie Universitaet Berlin, 14163 Berlin, Germany.
Graduate Research Training Program PharMetrX, 12169 Berlin, Germany.

Lena Klopp-Schulze (L)

Department of Clinical Pharmacy and Biochemistry, Institute of Pharmacy, Freie Universitaet Berlin, 14163 Berlin, Germany.

Robin Michelet (R)

Department of Clinical Pharmacy and Biochemistry, Institute of Pharmacy, Freie Universitaet Berlin, 14163 Berlin, Germany.

Madelé van Dyk (M)

College of Medicine and Public Health, Flinders University, Adelaide, SA 5042, Australia.

Thomas E Mürdter (TE)

Dr. Margarete Fischer-Bosch Institute of Clinical Pharmacology, Stuttgart, and University Tübingen, 70376 Tübingen, Germany.

Matthias Schwab (M)

Dr. Margarete Fischer-Bosch Institute of Clinical Pharmacology, 70376 Stuttgart, Germany.
German Cancer Consortium (DKTK), Partner Site Tübingen, German Cancer Research, 69120 Heidelberg, Germany.
Departments of Clinical Pharmacology, Pharmacy and Biochemistry, University Tübingen, 72076 Tübingen, Germany.

Markus Joerger (M)

Department of Medical Oncology and Hematology, Cantonal Hospital, 9007 St. Gallen, Switzerland.

Wilhelm Huisinga (W)

Institute of Mathematics, University of Potsdam, 14476 Potsdam, Germany.

Gerd Mikus (G)

Department of Clinical Pharmacy and Biochemistry, Institute of Pharmacy, Freie Universitaet Berlin, 14163 Berlin, Germany.

Charlotte Kloft (C)

Department of Clinical Pharmacy and Biochemistry, Institute of Pharmacy, Freie Universitaet Berlin, 14163 Berlin, Germany.

Classifications MeSH