In Vitro Effects of Low Doses of β-Caryophyllene, Ascorbic Acid and d-Glucosamine on Human Chondrocyte Viability and Inflammation.

ascorbic acid chondrocyte d-glucosamine inflammation osteoarthritis reactive oxygen species β-caryophyllene

Journal

Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453

Informations de publication

Date de publication:
23 Mar 2021
Historique:
received: 08 02 2021
revised: 13 03 2021
accepted: 20 03 2021
entrez: 3 4 2021
pubmed: 4 4 2021
medline: 4 4 2021
Statut: epublish

Résumé

β-caryophyllene (BCP), a plant-derived sesquiterpene, has been reported to have anti-inflammatory and antioxidant effects. The purpose of this study is to evaluate the effects of BCP in combination with ascorbic acid (AA) and d-glucosamine (GlcN) against macrophage-mediated inflammation on in vitro primary human chondrocytes. Changes in cell viability, intracellular ROS generation, gene expression of pro-inflammatory mediators, metalloproteinases (MMPs), collagen type II and aggrecan were analyzed in primary human chondrocytes exposed to the conditioned medium (CM) of activated U937 monocytes and subsequently treated with BCP alone or in combination with AA and GlcN. The CM-induced chondrocyte cytotoxicity was reduced by the presence of low doses of BCP alone or in combination with AA and GlcN. The exposure of cells to CM significantly increased

Identifiants

pubmed: 33806983
pii: ph14030286
doi: 10.3390/ph14030286
pmc: PMC8005039
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : UNI-Impresa, University of Padova, Italy
ID : 0

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Auteurs

Elena Mattiuzzo (E)

Department of Molecular Medicine, Histology Unit, University of Padova, 35121 Padova, Italy.

Alessia Faggian (A)

Department of Molecular Medicine, Histology Unit, University of Padova, 35121 Padova, Italy.

Rina Venerando (R)

Department of Molecular Medicine, University of Padova, 35121 Padova, Italy.

Andrea Benetti (A)

Department of Molecular Medicine, Histology Unit, University of Padova, 35121 Padova, Italy.

Elisa Belluzzi (E)

Musculoskeletal Pathology and Oncology Laboratory, Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.
Orthopaedic and Traumatology Clinic, Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.

Giovanni Abatangelo (G)

Faculty of Medicine, University of Padova, 35100 Padova, Italy.

Pietro Ruggieri (P)

Orthopaedic and Traumatology Clinic, Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.

Paola Brun (P)

Department of Molecular Medicine, Histology Unit, University of Padova, 35121 Padova, Italy.

Classifications MeSH