Dispirooxindoles Based on 2-Selenoxo-Imidazolidin-4-Ones: Synthesis, Cytotoxicity and ROS Generation Ability.


Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
05 Mar 2021
Historique:
received: 13 12 2020
revised: 25 02 2021
accepted: 01 03 2021
entrez: 3 4 2021
pubmed: 4 4 2021
medline: 23 4 2021
Statut: epublish

Résumé

A regio- and diastereoselective synthesis of two types of dispiro derivatives of 2-selenoxoimidazolidin-4-ones, differing in the position of the nitrogen atom in the central pyrrolidine ring of the spiro-fused system-namely, 2-selenoxodispiro[imidazolidine-4,3'-pyrrolidine-2',3″-indoline]-2″,5-diones (

Identifiants

pubmed: 33807662
pii: ijms22052613
doi: 10.3390/ijms22052613
pmc: PMC7961907
pii:
doi:

Substances chimiques

Cytotoxins 0
Pyrrolidines 0
Reactive Oxygen Species 0
TP53 protein, human 0
Tumor Suppressor Protein p53 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Russian Foundation for Basic Research
ID : 19-03-00201
Organisme : Russian Foundation for Basic Research
ID : 20-33-90008
Organisme : Russian Science Foundation
ID : 19-79-30062
Organisme : Competitiveness Program of NUST "MISIS"
ID : Governmental decree dated March 16, 2013, No. 211

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Auteurs

Vladimir K Novotortsev (VK)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

Maxim E Kukushkin (ME)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.

Viktor A Tafeenko (VA)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

Dmitry A Skvortsov (DA)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

Marina A Kalinina (MA)

Skolkovo Institute of Science and Technology, 4 Alfred Nobel Street, Skolkovo, 143025 Moscow, Russia.

Roman V Timoshenko (RV)

National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.

Nelly S Chmelyuk (NS)

National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.

Liliya A Vasilyeva (LA)

Faculty of Bioengineering and Bioinformatics, Lomonosov Moscow State University, Leninskie Gory 1, 119991 Moscow, Russia.

Boris N Tarasevich (BN)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

Petr V Gorelkin (PV)

National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.

Alexander S Erofeev (AS)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.

Alexander G Majouga (AG)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
National University of Science and Technology "MISiS", Leninskiy Prospect, 4, 119049 Moscow, Russia.
D. I. Mendeleev University of Chemical Technology of Russia, Miusskaya sq., 9, 125047 Moscow, Russia.

Nikolai V Zyk (NV)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

Elena K Beloglazkina (EK)

Department of Chemistry, M. V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.

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Classifications MeSH