Diaryl Ureas as an Antiprotozoal Chemotype.

Animals Antiprotozoal Agents / pharmacology Leishmania donovani Mice Trypanosoma brucei rhodesiense Trypanosoma cruzi Urea
N,N′-diarylurea antiprotozoal chemotype

Journal

ACS infectious diseases
ISSN: 2373-8227
Titre abrégé: ACS Infect Dis
Pays: United States
ID NLM: 101654580

Informations de publication

Date de publication:
11 06 2021
Historique:
pubmed: 11 5 2021
medline: 24 6 2021
entrez: 10 5 2021
Statut: ppublish

Résumé

We now describe the physicochemical profiling,

Identifiants

DOI: 10.1021/acsinfecdis.1c00135 PMID: 33971090 PMC: PMC8802619
pubmed: 33971090
doi: 10.1021/acsinfecdis.1c00135
pmc: PMC8802619
mid: NIHMS1771891
doi:

Substances chimiques

Antiprotozoal Agents 0
Urea 8W8T17847W

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

1578-1583

Subventions

Organisme : NIGMS NIH HHS
ID : P20 GM103427
Pays : United States
Organisme : NIAID NIH HHS
ID : R01 AI116723
Pays : United States

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Auteurs

Derek A Leas (DA)

College of Pharmacy, University of Nebraska Medical Center, 986125 Nebraska Medical Center, Omaha, Nebraska 68198-6125, United States.

Austin G Sanford (AG)

Department of Pathology & Microbiology, College of Medicine, University of Nebraska Medical Center, 985900 Nebraska Medical Center, Omaha, Nebraska 68198-5900, United States.
Department of Biology, University of Nebraska at Omaha, 6001 Dodge Street, Omaha, Nebraska 68182, United States.

Jianbo Wu (J)

College of Pharmacy, University of Nebraska Medical Center, 986125 Nebraska Medical Center, Omaha, Nebraska 68198-6125, United States.

Monica Cal (M)

University of Basel, CH-4003 Basel, Switzerland.
Department of Medical Parasitology and Infection Biology, Swiss Tropical and Public Health Institute, CH-4002 Basel, Switzerland.

Marcel Kaiser (M)

University of Basel, CH-4003 Basel, Switzerland.
Department of Medical Parasitology and Infection Biology, Swiss Tropical and Public Health Institute, CH-4002 Basel, Switzerland.

Sergio Wittlin (S)

University of Basel, CH-4003 Basel, Switzerland.
Department of Medical Parasitology and Infection Biology, Swiss Tropical and Public Health Institute, CH-4002 Basel, Switzerland.

Ryan M Hemsley (RM)

Department of Biology, University of Nebraska at Omaha, 6001 Dodge Street, Omaha, Nebraska 68182, United States.

Elyssa B Darner (EB)

Department of Biology, University of Nebraska at Omaha, 6001 Dodge Street, Omaha, Nebraska 68182, United States.

LeeAnna M Lui (LM)

Department of Biology, University of Nebraska at Omaha, 6001 Dodge Street, Omaha, Nebraska 68182, United States.

Paul H Davis (PH)

Department of Biology, University of Nebraska at Omaha, 6001 Dodge Street, Omaha, Nebraska 68182, United States.
ORCID: 0000-0002-0526-3841

Jonathan L Vennerstrom (JL)

College of Pharmacy, University of Nebraska Medical Center, 986125 Nebraska Medical Center, Omaha, Nebraska 68198-6125, United States.
ORCID: 0000-0003-0075-2336

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Classifications MeSH

questionsmedicales.fr › Eucaryotes › Animaux › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Actions chimiques et utilisations › Actions pharmacologiques › Utilisations thérapeutiques › Anti-infectieux › Antiparasitaires › Antiprotozoaires › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Eucaryotes › Euglénozoaires › Kinetoplastida › Trypanosomatina › Leishmania › Leishmania donovani › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Rodentia › Muridae › Murinae › Souris › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Eucaryotes › Euglénozoaires › Kinetoplastida › Trypanosomatina › Trypanosoma › Trypanosoma brucei rhodesiense › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Eucaryotes › Euglénozoaires › Kinetoplastida › Trypanosomatina › Trypanosoma › Trypanosoma cruzi › Diaryl Ureas as an Antiprotozoal Chemotype.
questionsmedicales.fr › Composés chimiques organiques › Amides › Urée › Diaryl Ureas as an Antiprotozoal Chemotype.