Flavin-Helicene Amphiphilic Hybrids: Synthesis, Characterization, and Preparation of Surface-Supported Films.

flavins helicenes lipidic cubic phases redox behavior thin layers

Journal

ChemPlusChem
ISSN: 2192-6506
Titre abrégé: Chempluschem
Pays: Germany
ID NLM: 101580948

Informations de publication

Date de publication:
11 May 2021
Historique:
revised: 20 04 2021
received: 25 02 2021
pubmed: 13 5 2021
medline: 13 5 2021
entrez: 12 5 2021
Statut: aheadofprint

Résumé

This work reports on the preparation and structural characterization of flavo[7]helicene 1 (flavin-[7]helicene conjugate), which was subsequently characterized at the molecular level in either an aqueous environment or an organic phase, at the supramolecular level in the form of polymeric layers, and also embedded in a lipidic mesophase environment to study the resulting properties of such a hybrid relative to its parent molecules. The flavin benzo[g]pteridin-2,4-dione (isoalloxazine) was selected for conjugation because of its photoactivity and reversible redox behavior. Compound 1 was prepared from 2-nitroso[6]helicene and 6-methylamino-3-methyluracil, and characterized using common structural and spectroscopic tools: circular dichroism (CD), circularly polarized luminescence (CPL) spectroscopy, cyclic voltammetry (CV), and DFT quantum calculations. In addition, a methodology that allows the loading of 1 enantiomers into an internally nanostructured lipid (1-monoolein) matrix was developed.

Identifiants

pubmed: 33977667
doi: 10.1002/cplu.202100092
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

982-990

Subventions

Organisme : Institute of Chemical Process Fundamentals of the CAS
Organisme : Palacky University
ID : RVO 61989592
Organisme : Palacky University
ID : IGA_LF_2020_022
Organisme : Ministry of Education, Youth and Sports
Organisme : Czech Science Foundation
ID : 20-19353S
Organisme : Czech Science Foundation
ID : CZ.02.2.69/0.0/0.0/16_027/0008482
Organisme : Czech Science Foundation
ID : e-INFRA LM2018140

Informations de copyright

© 2021 Wiley-VCH GmbH.

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Auteurs

Martin Jakubec (M)

Institute of Chemical Process Fundamentals of the Czech Academy of Sciences, v.v.i., Rozvojová 135, 165 02, Prague 6, Czech Republic.

David Novák (D)

Department of Medical Chemistry and Biochemistry, Faculty of Medicine and Dentistry, Palacký University, Hněvotínská 3, 775 15, Olomouc, Czech Republic.

Martina Zatloukalová (M)

Department of Medical Chemistry and Biochemistry, Faculty of Medicine and Dentistry, Palacký University, Hněvotínská 3, 775 15, Olomouc, Czech Republic.

Ivana Císařová (I)

Department of Inorganic Chemistry, Faculty of Science, Charles University in Prague, Hlavova 2030, 128 40, Prague 2, Czech Republic.

Radek Cibulka (R)

Department of Organic Chemistry, University of Chemistry and Technology, Prague, Technická 5, 166 28, Prague, Czech Republic.

Ludovic Favereau (L)

Univ. Rennes, CNRS, ISCR-UMR 6226, Campus de Beaulieu, 35042, Rennes Cedex, France.

Jeanne Crassous (J)

Univ. Rennes, CNRS, ISCR-UMR 6226, Campus de Beaulieu, 35042, Rennes Cedex, France.

Adrianna Cytryniak (A)

Faculty of Chemistry, University of Warsaw, Pasteura 1, Warsaw, 02-093, Poland.

Renata Bilewicz (R)

Faculty of Chemistry, University of Warsaw, Pasteura 1, Warsaw, 02-093, Poland.

Jan Hrbáč (J)

Institute of Chemistry, Masaryk University, Kamenice 5, Brno, 725 00, Czech Republic.

Jan Storch (J)

Institute of Chemical Process Fundamentals of the Czech Academy of Sciences, v.v.i., Rozvojová 135, 165 02, Prague 6, Czech Republic.

Jaroslav Žádný (J)

Institute of Chemical Process Fundamentals of the Czech Academy of Sciences, v.v.i., Rozvojová 135, 165 02, Prague 6, Czech Republic.

Jan Vacek (J)

Department of Medical Chemistry and Biochemistry, Faculty of Medicine and Dentistry, Palacký University, Hněvotínská 3, 775 15, Olomouc, Czech Republic.

Classifications MeSH