PPARγ induces PD-L1 expression in MSS+ colorectal cancer cells.


Journal

Oncoimmunology
ISSN: 2162-402X
Titre abrégé: Oncoimmunology
Pays: United States
ID NLM: 101570526

Informations de publication

Date de publication:
05 05 2021
Historique:
entrez: 24 5 2021
pubmed: 25 5 2021
medline: 3 8 2021
Statut: epublish

Résumé

Only a small subset of colorectal cancer (CRC) patients benefits from immunotherapies, comprising blocking antibodies (Abs) against checkpoint receptor "programmed-cell-death-1" (PD1) and its ligand (PD-L1), because most cases lack the required mutational burden and neo-antigen load caused by microsatellite instability (MSI) and/or an inflamed, immune cell-infiltrated PD-L1+ tumor microenvironment. Peroxisome proliferator-activated-receptor-gamma (PPARγ), a metabolic transcription factor stimulated by anti-diabetic drugs, has been previously implicated in pre/clinical responses to immunotherapy. We therefore raised the hypothesis that PPARγ induces PD-L1 on microsatellite stable (MSS) tumor cells to enhance Ab-target engagement and responsiveness to PD-L1 blockage. We found that PPARγ-agonists upregulate PD-L1 mRNA/protein expression in human gastrointestinal cancer cell lines and MSS+ patient-derived tumor organoids (PDOs). Mechanistically, PPARγ bound to and activated DNA-motifs similar to cognate PPARγ-responsive-elements (PPREs) in the proximal -2 kb promoter of the human

Identifiants

pubmed: 34026331
doi: 10.1080/2162402X.2021.1906500
pii: 1906500
pmc: PMC8115557
doi:

Substances chimiques

B7-H1 Antigen 0
PPAR gamma 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1906500

Informations de copyright

© 2021 The Author(s). Published with license by Taylor & Francis Group, LLC.

Références

J Clin Oncol. 2018 Oct 25;:JCO1800632
pubmed: 30359157
Immun Inflamm Dis. 2020 Mar;8(1):8-23
pubmed: 31742928
Ann Oncol. 2019 Jul 1;30(7):1134-1142
pubmed: 30918950
Pathologe. 2018 Nov;39(6):498-519
pubmed: 30367225
Immunity. 2018 Jan 16;48(1):147-160.e7
pubmed: 29343435
Nat Commun. 2017 Oct 3;8(1):766
pubmed: 28974683
J Clin Invest. 2017 Aug 1;127(8):2930-2940
pubmed: 28650338
Nat Immunol. 2018 Dec;19(12):1330-1340
pubmed: 30420624
Nat Rev Endocrinol. 2017 Jan;13(1):36-49
pubmed: 27636730
Nat Med. 2015 Nov;21(11):1350-6
pubmed: 26457759
Metabolism. 2013 Jun;62(6):778-85
pubmed: 23398844
Blood. 2004 Nov 15;104(10):3276-84
pubmed: 15265789
J Immunother Cancer. 2019 Feb 27;7(1):57
pubmed: 30813970
Cancer Immunol Res. 2018 Jun;6(6):723-732
pubmed: 29669721
N Engl J Med. 2012 Apr 5;366(14):1345-7
pubmed: 22475600
N Engl J Med. 2015 Jun 25;372(26):2509-20
pubmed: 26028255
Mol Cell. 1999 Jun;3(6):799-804
pubmed: 10394368
Leuk Lymphoma. 2003 Sep;44(9):1457-62
pubmed: 14565644
Immunity. 2016 Aug 16;45(2):358-73
pubmed: 27496729
Blood. 2006 Jul 15;108(2):525-35
pubmed: 16527895
Nat Commun. 2017 Jul 24;8(1):103
pubmed: 28740126
Nat Med. 2018 Mar;24(3):360-367
pubmed: 29377004
Oncoimmunology. 2018 Aug 23;7(11):e1500107
pubmed: 30393583
J Exp Med. 2018 Apr 2;215(4):1091-1100
pubmed: 29511066
J Surg Res. 2012 May 1;174(1):1-6
pubmed: 21816436
Nature. 2015 Sep 17;525(7569):380-3
pubmed: 26331539
Oncotarget. 2016 Sep 27;7(39):63093-63105
pubmed: 27494857
Cell. 2018 Sep 6;174(6):1586-1598.e12
pubmed: 30100188
Proc Natl Acad Sci U S A. 2017 Jan 31;114(5):E761-E770
pubmed: 28096382
Nat Rev Clin Oncol. 2019 Sep;16(9):563-580
pubmed: 31092901
Immunity. 2016 Mar 15;44(3):698-711
pubmed: 26982367
Nature. 2012 Jun 28;486(7404):549-53
pubmed: 22722857
Science. 2018 Oct 12;362(6411):
pubmed: 30309915
Semin Cancer Biol. 2019 Apr;55:78-89
pubmed: 29716829
Nat Rev Gastroenterol Hepatol. 2018 Dec;15(12):721-737
pubmed: 30185915
Nat Rev Cancer. 2012 Feb 09;12(3):181-95
pubmed: 22318237
JAMA Oncol. 2020 Apr 1;6(4):512-518
pubmed: 31876896
Cancer Immunol Immunother. 2017 Jul;66(7):927-939
pubmed: 28405764
Cancer Res Treat. 2019 Jun 12;:
pubmed: 31208164
Cancer Cell. 2019 Aug 12;36(2):168-178.e4
pubmed: 31327656
Cancer Immunol Res. 2018 Nov;6(11):1375-1387
pubmed: 30143538
Nat Med. 2019 Jan;25(1):141-151
pubmed: 30420753
Cancer Immunol Res. 2019 Oct;7(10):1570-1573
pubmed: 31405947
Nat Cell Biol. 2017 Nov;19(11):1336-1347
pubmed: 29035359
Nat Commun. 2019 May 16;10(1):2197
pubmed: 31097693
Cell Rep. 2017 May 9;19(6):1189-1201
pubmed: 28494868
Cancer Immunol Res. 2016 Jul;4(7):563-8
pubmed: 27197067
J Heart Lung Transplant. 2011 Jun;30(6):698-706
pubmed: 21435906
Oncol Lett. 2019 Dec;18(6):5977-5985
pubmed: 31788072
Cell. 2019 Sep 19;179(1):236-250.e18
pubmed: 31495571
Science. 2019 Jun 07;364(6444):952-955
pubmed: 31171691
PPAR Res. 2008;2008:309469
pubmed: 18596912
Blood. 2012 Jan 5;119(1):115-26
pubmed: 22053106
J Cancer Res Ther. 2018 Jun;14(Supplement):S306-S310
pubmed: 29970681
Cell. 2018 Dec 13;175(7):1972-1988.e16
pubmed: 30550791
Clin Cancer Res. 2016 Aug 15;22(16):4057-66
pubmed: 26994146
Immunol Rev. 2017 Mar;276(1):112-120
pubmed: 28258695
Mol Cell Biol. 2011 Aug;31(16):3497-510
pubmed: 21690289
Lancet Oncol. 2019 Jun;20(6):849-861
pubmed: 31003911
Science. 2018 Feb 23;359(6378):920-926
pubmed: 29472484
Cancer Cell. 2017 Sep 11;32(3):377-391.e9
pubmed: 28898698

Auteurs

Tobias Gutting (T)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Veronika Hauber (V)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Jens Pahl (J)

Department of Immunobiochemistry, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Mannheim Institute for Innate Immunoscience (MI3), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Kay Klapproth (K)

Department of Immunobiochemistry, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Mannheim Institute for Innate Immunoscience (MI3), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Wenyue Wu (W)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Department of Immunobiochemistry, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Ioana Dobrota (I)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Department of Immunobiochemistry, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Frank Herweck (F)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Juliane Reichling (J)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Laura Helm (L)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Torsten Schroeder (T)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Beifang Li (B)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Philip Weidner (P)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Tianzuo Zhan (T)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Maximilian Eckardt (M)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Johannes Betge (J)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Junior Clinical Cooperation Unit Translational Gastrointestinal Oncology and Preclinical Models (B440), German Cancer Research Center (DKFZ), Heidelberg, Germany.

Sebastian Belle (S)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Carsten Sticht (C)

Center for Medical Research (ZMF), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Timo Gaiser (T)

Institute of Pathology, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Michael Boutros (M)

Division Signaling and Functional Genomics, German Cancer Research Center (DKFZ) and Heidelberg University, Heidelberg, Germany.

Matthias P A Ebert (MPA)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Mannheim Institute for Innate Immunoscience (MI3), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
European Center of Angioscience (ECAS), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Adelheid Cerwenka (A)

Department of Immunobiochemistry, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Mannheim Institute for Innate Immunoscience (MI3), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
European Center of Angioscience (ECAS), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Elke Burgermeister (E)

Department of Medicine II, University Medical Center Mannheim, Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.
Mannheim Institute for Innate Immunoscience (MI3), Medical Faculty Mannheim, Heidelberg University, Mannheim, Germany.

Articles similaires

[Redispensing of expensive oral anticancer medicines: a practical application].

Lisanne N van Merendonk, Kübra Akgöl, Bastiaan Nuijen
1.00
Humans Antineoplastic Agents Administration, Oral Drug Costs Counterfeit Drugs

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH