Toward New Transmission-Blocking Combination Therapies: Pharmacokinetics of 10-Amino-Artemisinins and 11-Aza-Artemisinin and Comparison with Dihydroartemisinin and Artemether.
amino-artemisinins
antimalarial agents
combination therapies
pharmacokinetics
transmission-blocking
Journal
Antimicrobial agents and chemotherapy
ISSN: 1098-6596
Titre abrégé: Antimicrob Agents Chemother
Pays: United States
ID NLM: 0315061
Informations de publication
Date de publication:
16 07 2021
16 07 2021
Historique:
pubmed:
8
6
2021
medline:
10
8
2021
entrez:
7
6
2021
Statut:
ppublish
Résumé
As artemisinin combination therapies (ACTs) are compromised by resistance, we are evaluating triple combination therapies (TACTs) comprising an amino-artemisinin, a redox drug, and a third drug with a different mode of action. Thus, here we briefly review efficacy data on artemisone, artemiside, other amino-artemisinins, and 11-aza-artemisinin and conduct absorption, distribution, and metabolism and excretion (ADME) profiling
Identifiants
pubmed: 34097488
doi: 10.1128/AAC.00990-21
pmc: PMC8284440
doi:
Substances chimiques
Antimalarials
0
Artemisinins
0
artenimol
6A9O50735X
Artemether
C7D6T3H22J
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
e0099021Références
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