Novel antibody cocktail targeting Bet v 1 rapidly and sustainably treats birch allergy symptoms in a phase 1 study.


Journal

The Journal of allergy and clinical immunology
ISSN: 1097-6825
Titre abrégé: J Allergy Clin Immunol
Pays: United States
ID NLM: 1275002

Informations de publication

Date de publication:
01 2022
Historique:
received: 01 02 2021
revised: 06 05 2021
accepted: 14 05 2021
pubmed: 15 6 2021
medline: 4 3 2022
entrez: 14 6 2021
Statut: ppublish

Résumé

The efficacy of an allergen-specific IgG cocktail to treat cat allergy suggests that allergen-specific IgG may be a major protective mechanism elicited by allergen immunotherapy. Extending these findings, we tested a Bet v 1-specific antibody cocktail in birch-allergic subjects. This was a phase 1, randomized, double-blind, study with 2 parts. Part A administered ascending doses of the Bet v 1-specific antibody cocktail REGN5713/14/15 (150-900 mg) in 32 healthy adults. Part B administered a single subcutaneous 900-mg dose or placebo in 64 birch-allergic subjects. Total nasal symptom score response to titrated birch extract nasal allergen challenge and skin prick test (SPT) with birch and alder allergen were assessed at screening and days 8, 29, 57, and 113 (SPT only); basophil activation tests (n = 26) were conducted. Single-dose REGN5713/14/15 significantly reduced total nasal symptom score following birch nasal allergen challenge relative to baseline. Differences in total nasal symptom score areas under the curve (0-1 hour) for subjects treated with REGN5713/14/15 versus those given placebo (day 8: -1.17, P = .001; day 29: -1.18, P = .001; day 57: -0.85, P = .024) and titration SPT with birch difference in area under the curve of mean wheal diameters for subjects treated with REGN5713/14/15 versus placebo (all P < .001) were sustained for ≥2 months; similar results were observed with alder SPT. REGN5713/14/15 was well tolerated. Basophil responsiveness to birch-related allergens was significantly decreased in subjects treated with REGN5713/14/15 versus those given placebo on days 8, 57, and 113 (all P < .01). Single-dose REGN5713/14/15 was well tolerated and provided a rapid (1 week) and durable (2 months) reduction in allergic symptoms after birch allergen nasal allergen challenge, potentially offering a new paradigm for the treatment of birch allergy symptoms.

Sections du résumé

BACKGROUND
The efficacy of an allergen-specific IgG cocktail to treat cat allergy suggests that allergen-specific IgG may be a major protective mechanism elicited by allergen immunotherapy.
OBJECTIVES
Extending these findings, we tested a Bet v 1-specific antibody cocktail in birch-allergic subjects.
METHODS
This was a phase 1, randomized, double-blind, study with 2 parts. Part A administered ascending doses of the Bet v 1-specific antibody cocktail REGN5713/14/15 (150-900 mg) in 32 healthy adults. Part B administered a single subcutaneous 900-mg dose or placebo in 64 birch-allergic subjects. Total nasal symptom score response to titrated birch extract nasal allergen challenge and skin prick test (SPT) with birch and alder allergen were assessed at screening and days 8, 29, 57, and 113 (SPT only); basophil activation tests (n = 26) were conducted.
RESULTS
Single-dose REGN5713/14/15 significantly reduced total nasal symptom score following birch nasal allergen challenge relative to baseline. Differences in total nasal symptom score areas under the curve (0-1 hour) for subjects treated with REGN5713/14/15 versus those given placebo (day 8: -1.17, P = .001; day 29: -1.18, P = .001; day 57: -0.85, P = .024) and titration SPT with birch difference in area under the curve of mean wheal diameters for subjects treated with REGN5713/14/15 versus placebo (all P < .001) were sustained for ≥2 months; similar results were observed with alder SPT. REGN5713/14/15 was well tolerated. Basophil responsiveness to birch-related allergens was significantly decreased in subjects treated with REGN5713/14/15 versus those given placebo on days 8, 57, and 113 (all P < .01).
CONCLUSIONS
Single-dose REGN5713/14/15 was well tolerated and provided a rapid (1 week) and durable (2 months) reduction in allergic symptoms after birch allergen nasal allergen challenge, potentially offering a new paradigm for the treatment of birch allergy symptoms.

Identifiants

pubmed: 34126156
pii: S0091-6749(21)00904-0
doi: 10.1016/j.jaci.2021.05.039
pii:
doi:

Substances chimiques

Allergens 0
Antibodies, Monoclonal 0
Antigens, Plant 0
Immunoglobulin G 0
Bet v 1 allergen, Betula 126161-14-6

Banques de données

ClinicalTrials.gov
['NCT03969849']

Types de publication

Clinical Trial, Phase I Journal Article Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

189-199

Informations de copyright

Copyright © 2021 The Authors. Published by Elsevier Inc. All rights reserved.

Auteurs

Philippe Gevaert (P)

Department of Otorhinolaryngology, Ghent University Hospital, Ghent, Belgium.

Jarno De Craemer (J)

Department of Otorhinolaryngology, Ghent University Hospital, Ghent, Belgium.

Natalie De Ruyck (N)

Department of Otorhinolaryngology, Ghent University Hospital, Ghent, Belgium.

Sylvie Rottey (S)

Drug Research Unit Ghent, Ghent University Hospital, Ghent, Belgium.

Jan de Hoon (J)

Center for Clinical Pharmacology, UZ Leuven, Leuven, Belgium.

Peter W Hellings (PW)

Department of Otorhinolaryngology, Ghent University Hospital, Ghent, Belgium; Allergy and Clinical Immunology Research Group, KU Leuven, Leuven, Belgium; Academic Medical Center Amsterdam, University of Amsterdam, Amsterdam, The Netherlands.

Bram Volckaert (B)

SGS Belgium Clinical Pharmacology Unit Antwerpen, Antwerp, Belgium.

Kristof Lesneuck (K)

SGS Belgium Clinical Pharmacology Unit Antwerpen, Antwerp, Belgium.

Jamie M Orengo (JM)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Amanda Atanasio (A)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Mohamed A Kamal (MA)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Hisham Abdallah (H)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Vishal Kamat (V)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Robert Dingman (R)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Michelle DeVeaux (M)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Divya Ramesh (D)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Lorah Perlee (L)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Claire Q Wang (CQ)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

David M Weinreich (DM)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Gary Herman (G)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

George D Yancopoulos (GD)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY.

Meagan P O'Brien (MP)

Regeneron Pharmaceuticals, Inc, Tarrytown, NY. Electronic address: meagan.obrien@regeneron.com.

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Classifications MeSH