Evaluation of Benzguinols as Next-Generation Antibiotics for the Treatment of Multidrug-Resistant Bacterial Infections.
Gram-negative
Staphylococcus aureus
Staphylococcus pseudintermedius
antimicrobial resistance
benzguinols
bioluminescent mouse model
colistin
cytotoxicity
minimum inhibitory concentration
nidulins
Journal
Antibiotics (Basel, Switzerland)
ISSN: 2079-6382
Titre abrégé: Antibiotics (Basel)
Pays: Switzerland
ID NLM: 101637404
Informations de publication
Date de publication:
16 Jun 2021
16 Jun 2021
Historique:
received:
12
05
2021
revised:
10
06
2021
accepted:
10
06
2021
entrez:
2
7
2021
pubmed:
3
7
2021
medline:
3
7
2021
Statut:
epublish
Résumé
Our recent focus on the "lost antibiotic" unguinol and related nidulin-family fungal natural products identified two semisynthetic derivatives, benzguinols A and B, with unexpected in vitro activity against
Identifiants
pubmed: 34208698
pii: antibiotics10060727
doi: 10.3390/antibiotics10060727
pmc: PMC8233939
pii:
doi:
Types de publication
Journal Article
Langues
eng
Subventions
Organisme : Cooperative Research Centres, Australian Government Department of Industry
ID : CRCPFIVE000119
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