Photochemical (Hetero-)Arylation of Aryl Sulfonium Salts.


Journal

Organic letters
ISSN: 1523-7052
Titre abrégé: Org Lett
Pays: United States
ID NLM: 100890393

Informations de publication

Date de publication:
20 08 2021
Historique:
pubmed: 31 7 2021
medline: 31 7 2021
entrez: 30 7 2021
Statut: ppublish

Résumé

The construction of (hetero)biaryls, which are ubiquitous scaffolds among medical substances, functional materials, and agrochemicals, constitutes a key application of cross-coupling methods. However, these usually require multiple synthetic steps. Herein, we report a simple photoinduced and catalyst-free C-H/C-H (hetero)arylation cross-coupling through aryl thianthrenium salts, which are formed site-selectively by direct C-H functionalization. The key to this approach is the UV-light, which can disrupt the C-S bond to form thianthrene radical cations and aryl radicals.

Identifiants

pubmed: 34327991
doi: 10.1021/acs.orglett.1c01904
pmc: PMC8383302
doi:

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

6232-6236

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Auteurs

Yue Zhao (Y)

Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, 52074 Aachen, Germany.

Congjun Yu (C)

Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, 52074 Aachen, Germany.

Wenjing Liang (W)

Institute of Physical Chemistry, RWTH Aachen University, Landoltweg 1, 52074 Aachen, Germany.

Frederic W Patureau (FW)

Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, 52074 Aachen, Germany.

Classifications MeSH