Machine Learning Models Identify Inhibitors of SARS-CoV-2.


Journal

Journal of chemical information and modeling
ISSN: 1549-960X
Titre abrégé: J Chem Inf Model
Pays: United States
ID NLM: 101230060

Informations de publication

Date de publication:
27 09 2021
Historique:
pubmed: 14 8 2021
medline: 30 9 2021
entrez: 13 8 2021
Statut: ppublish

Résumé

With the rapidly evolving SARS-CoV-2 variants of concern, there is an urgent need for the discovery of further treatments for the coronavirus disease (COVID-19). Drug repurposing is one of the most rapid strategies for addressing this need, and numerous compounds have already been selected for

Identifiants

pubmed: 34387990
doi: 10.1021/acs.jcim.1c00683
pmc: PMC8574161
mid: NIHMS1750561
doi:

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

4224-4235

Subventions

Organisme : NIGMS NIH HHS
ID : R44 GM122196
Pays : United States
Organisme : NCCIH NIH HHS
ID : R43 AT010585
Pays : United States

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Auteurs

Victor O Gawriljuk (VO)

São Carlos Institute of Physics, University of São Paulo, Av. João Dagnone, 1100-Santa Angelina, São Carlos, São Paulo 13563-120, Brazil.

Phyo Phyo Kyaw Zin (PPK)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

Ana C Puhl (AC)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

Kimberley M Zorn (KM)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

Daniel H Foil (DH)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

Thomas R Lane (TR)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

Brett Hurst (B)

Institute for Antiviral Research, Utah State University, Logan, Utah 84322-5600, United States.
Department of Animal, Dairy and Veterinary Sciences, Utah State University, Logan, Utah 84322-4815, United States.

Tatyana Almeida Tavella (TA)

Laboratory of Tropical Diseases-Prof. Dr. Luiz Jacinto da Silva, Department of Genetics, Evolution, Microbiology and Immunology, University of Campinas-UNICAMP, Campinas, São Paulo, Brazil.

Fabio Trindade Maranhão Costa (FTM)

Laboratory of Tropical Diseases-Prof. Dr. Luiz Jacinto da Silva, Department of Genetics, Evolution, Microbiology and Immunology, University of Campinas-UNICAMP, Campinas, São Paulo, Brazil.

Premkumar Lakshmanane (P)

Department of Microbiology and Immunology, University of North Carolina School of Medicine, Chapel Hill North Carolina 27599, United States.

Jean Bernatchez (J)

Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, San Diego, California 92093, United States.

Andre S Godoy (AS)

São Carlos Institute of Physics, University of São Paulo, Av. João Dagnone, 1100-Santa Angelina, São Carlos, São Paulo 13563-120, Brazil.

Glaucius Oliva (G)

São Carlos Institute of Physics, University of São Paulo, Av. João Dagnone, 1100-Santa Angelina, São Carlos, São Paulo 13563-120, Brazil.

Jair L Siqueira-Neto (JL)

Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, San Diego, California 92093, United States.

Peter B Madrid (PB)

SRI International, 333 Ravenswood Avenue, Menlo Park, California 94025, United States.

Sean Ekins (S)

Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States.

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Classifications MeSH