Photocatalyzed E→Z Contra-thermodynamic Isomerization of Vinyl Boronates with Binaphthol.

alkenes binaphthol boron isomerization photochemistry

Journal

Chemistry (Weinheim an der Bergstrasse, Germany)
ISSN: 1521-3765
Titre abrégé: Chemistry
Pays: Germany
ID NLM: 9513783

Informations de publication

Date de publication:
07 Oct 2021
Historique:
received: 13 07 2021
pubmed: 20 8 2021
medline: 20 8 2021
entrez: 19 8 2021
Statut: ppublish

Résumé

The photocatalytic contra-thermodynamic E→Z isomerization of vinyl boronates by using a binaphthol catalyst is disclosed. The reaction, based on the transient formation of a suitable chromophore with a BINOL derivative as the catalyst, allowed geometrical isomerization in good-to-excellent Z/E ratio and excellent-to-quantitative yields. The mechanism of this E→Z contra-thermodynamic isomerization was studied, and the formation of a transient chromophore species is suggested.

Identifiants

pubmed: 34411357
doi: 10.1002/chem.202102536
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

13966-13970

Informations de copyright

© 2021 Wiley-VCH GmbH.

Références

F. Yang, M. Zhu, J. Zhang, H. Zhou, MedChemComm 2018, 9, 201-211.
B. R. Smith, C. M. Eastman, J. T. Njardarson, J. Med. Chem. 2014, 57, 9764-9773.
 
A. J. J. Lennox, G. C. Lloyd-Jones, Chem. Soc. Rev. 2014, 43, 412-443;
R. Armstrong, V. Aggarwal, Synthesis 2017, 49, 3323-3336;
N. Miyaura, A. Suzuki, Chem. Rev. 1995, 95, 2457-2483;
S. Namirembe, J. P. Morken, Chem. Soc. Rev. 2019, 48, 3464-3474;
J. W. B. Fyfe, A. J. B. Watson, Chem 2017, 3, 31-55;
J. Carreras, A. Caballero, P. J. Pérez, Chem. Asian J. 2019, 14, 329-343;
L. Xu, S. Zhang, P. Li, Chem. Soc. Rev. 2015, 44, 8848-8858;
G. Duret, R. Quinlan, P. Bisseret, N. Blanchard, Chem. Sci. 2015, 6, 5366-5382.
S. D. Roughley, A. M. Jordan, J. Med. Chem. 2011, 54, 3451-3479.
 
J. V. Obligacion, P. J. Chirik, Nat. Chem. Rev. 2018, 2, 15-34;
K. Burgess, M. J. Ohlmeyer, Chem. Rev. 1991, 91, 1179-1191.
 
E. T. Kiesewetter, R. V. O′Brien, E. C. Yu, S. J. Meek, R. R. Schrock, A. H. Hoveyda, J. Am. Chem. Soc. 2013, 135, 6026-6029;
T.-J. Hu, G. Zhang, Y.-H. Chen, C.-G. Feng, G.-Q. Lin, J. Am. Chem. Soc. 2016, 138, 2897-2900;
C. Wang, T. Tobrman, Z. Xu, E.-I. Negishi, Org. Lett. 2009, 11, 4092-4095;
T. Ohmura, Y. Yamamoto, N. Miyaura, J. Am. Chem. Soc. 2000, 122, 4990-4991;
W. J. Jang, W. L. Lee, J. H. Moon, J. Y. Lee, J. Yun, Org. Lett. 2016, 18, 1390-1393;
J. R. Coombs, L. Zhang, J. P. Morken, Org. Lett. 2015, 17, 1708-1711.
For reviews, see:
D. H. Waldeck, Chem. Rev. 1991, 91, 415-436;
C. Dugave, L. Demange, Chem. Rev. 2003, 103, 2475-2532;
J. J. Molloy, T. Morack, R. Gilmour, Angew. Chem. Int. Ed. 2019, 58, 13654-13664;
Angew. Chem. 2019, 131, 13789-13800.
 
K. Singh, S. J. Staig, J. D. Weaver, J. Am. Chem. Soc. 2014, 136, 5275-5278;
C. Onneken, K. Bussmann, R. Gilmour, Angew. Chem. Int. Ed. 2020, 59, 330-334;
Angew. Chem. 2020, 132, 338-342;
S. I. Faßbender, J. J. Molloy, C. Mück-Lichtenfeld, R. Gilmour, Angew. Chem. Int. Ed. 2019, 58, 18619-18626;
Angew. Chem. 2019, 131, 18792-18799;
J. B. Metternich, R. Gilmour, J. Am. Chem. Soc. 2015, 137, 11254-11257;
J. B. Metternich, D. G. Artiukhin, M. C. Holland, M. von Bremen-Kühne, J. Neugebauer, R. Gilmour, J. Org. Chem. 2017, 82, 9955-9977;
K. Livingstone, M. Tenberge, F. Pape, C. G. Daniliuc, C. Jamieson, R. Gilmour, Org. Lett. 2019, 21, 9677-9680;
S. I. Faßbender, J. B. Metternich, R. Gilmour, Org. Lett. 2018, 20, 724-727;
M. R. Becker, T. Morack, J. Robertson, J. B. Metternich, C. Mück-Lichtenfeld, C. Daniliuc, G. A. Burley, R. Gilmour, Tetrahedron 2020, 76, 131198;
W. Cai, H. Fan, D. Ding, Y. Zhang, W. Wang, Chem. Commun. 2017, 53, 12918-12921;
H. Li, H. Chen, Y. Zhou, J. Huang, J. Yi, H. Zhao, W. Wang, L. Jing, Chem. Asian J. 2020, 15, 555-559;
J. Xu, N. Liu, H. Lv, C. He, Z. Liu, X. Shen, F. Cheng, B. Fan, Green Chem. 2020, 22, 2739-2743;
Y.-M. Huang, S.-M. Wang, J. Leng, B. Moku, C. Zhao, N. S. Alharbi, H.-L. Qin, Eur. J. Org. Chem. 2019, 4597-4603;
H. Zhang, Q. Xu, L. Yu, S. Yu, Eur. J. Org. Chem. 2020, 1472-1477;
P. Shu, H. Xu, L. Zhang, J. Li, H. Liu, Y. Luo, X. Yang, Z. Ju, Z. Xu, SynOpen 2019, 3, 103-107;
C. Cruché, W. Neiderer, S. K. Collins, ACS Catal. 2021, 11, 8829-8836.
J. J. Molloy, J. B. Metternich, C. G. Daniliuc, A. J. B. Watson, R. Gilmour, Angew. Chem. Int. Ed. 2018, 57, 3168-3172;
Angew. Chem. 2018, 130, 3222-3226.
J. J. Molloy, M. Schäfer, M. Wienhold, T. Morack, C. G. Daniliuc, R. Gilmour, Science 2020, 369, 302-306.
 
A. Nitelet, D. Thevenet, B. Schiavi, C. Hardouin, J. Fournier, R. Tamion, X. Pannecoucke, P. Jubault, T. Poisson, Chem. Eur. J. 2019, 25, 3262-3266;
M. Zhong, Y. Gagné, T. Hope, X. Pannecoucke, M. Frenette, P. Jubault, T. Poisson, Angew. Chem. Int. Ed. 2021, 60, 14498-14503;
Angew. Chem. 2021, 133, 14619-14624;
M. Aelterman, M. Sayes, P. Jubault, T. Poisson, Chem. Eur. J. 2021, 27, 8277-8282;
M. Zhong, X. Pannecoucke, P. Jubault, T. Poisson, Chem. Eur. J. 2021, 27, 11818-11822.
T. Brégent, J.-P. Bouillon, T. Poisson, Org. Lett. 2020, 22, 7688-7693.
C. Brenninger, J. D. Jolliffe, T. Bach, Angew. Chem. Int. Ed. 2018, 57, 14338-14349;
Angew. Chem. 2018, 130, 14536-14547.
See the Supporting Information for details.
L. Pitzer, F. Schäfers, F. Glorius, Angew. Chem. Int. Ed. 2019, 58, 8572-8576;
Angew. Chem. 2019, 131, 8660-8664.
 
A. Tlili, F. Toulgoat, T. Billard, Angew. Chem. Int. Ed. 2016, 55, 11726-11735;
Angew. Chem. 2016, 128, 11900-11909;
T. Besset, P. Jubault, X. Pannecoucke, T. Poisson, Org. Chem. Front. 2016, 3, 1004-1010.
D. M. Knapp, E. P. Gillis, M. D. Burke, J. Am. Chem. Soc. 2009, 131, 6961-6963.
H. Noguchi, K. Hojo, M. Suginome, J. Am. Chem. Soc. 2007, 129, 758-759.
 
D. S. Barnett, P. N. Moquist, S. E. Schaus, Angew. Chem. Int. Ed. 2009, 48, 8679-8682;
Angew. Chem. 2009, 121, 8835-8838;
S. Lou, P. N. Moquist, S. E. Schaus, J. Am. Chem. Soc. 2007, 129, 15398-15404.
For selected examples of E→Z isomerization involving singlet state species, see:
F. D. Lewis, J. E. Elbert, A. L. Upthagrove, P. D. Hale, J. Org. Chem. 1991, 56, 553-561;
F. D. Lewis, S. V. Barancyk, J. Am. Chem. Soc. 1989, 111, 8653-8661;
T. Ishigami, K. Nakazato, M. Uehara, T. Endo, Tetrahedron Lett. 1979, 20, 863-866, and ref. [8e].

Auteurs

Thibaud Brégent (T)

Normandie Université, INSA Rouen, UNIROUEN, CNRS, COBRA (UMR 6014), 76000, Rouen, France.

Jean-Philippe Bouillon (JP)

Normandie Université, INSA Rouen, UNIROUEN, CNRS, COBRA (UMR 6014), 76000, Rouen, France.

Thomas Poisson (T)

Normandie Université, INSA Rouen, UNIROUEN, CNRS, COBRA (UMR 6014), 76000, Rouen, France.
Institut Universitaire de France, 1 rue Descartes, 75231, Paris, France.

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