Review of Transporter Substrate, Inhibitor, and Inducer Characteristics of Cladribine.
Journal
Clinical pharmacokinetics
ISSN: 1179-1926
Titre abrégé: Clin Pharmacokinet
Pays: Switzerland
ID NLM: 7606849
Informations de publication
Date de publication:
12 2021
12 2021
Historique:
accepted:
28
07
2021
pubmed:
27
8
2021
medline:
28
1
2022
entrez:
26
8
2021
Statut:
ppublish
Résumé
Cladribine is a nucleoside analog that is phosphorylated in its target cells (B- and T-lymphocytes) to its active adenosine triphosphate form (2-chlorodeoxyadenosine triphosphate). Cladribine tablets 10 mg (Mavenclad
Identifiants
pubmed: 34435310
doi: 10.1007/s40262-021-01065-3
pii: 10.1007/s40262-021-01065-3
pmc: PMC8613159
doi:
Substances chimiques
ATP Binding Cassette Transporter, Subfamily G, Member 2
0
ATP-Binding Cassette Transporters
0
Membrane Transport Proteins
0
Neoplasm Proteins
0
Cladribine
47M74X9YT5
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Review
Langues
eng
Sous-ensembles de citation
IM
Pagination
1509-1535Subventions
Organisme : merck healthcare kgaa
ID : CrossRef Funder ID: 10.13039/100009945
Informations de copyright
© 2021. The Author(s).
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