Optimization and Evaluation of the In Vitro Permeation Parameters of Topical Products with Non-Steroidal Anti-Inflammatory Drugs through Strat-M
Plackett–Burman design
Strat-M® membrane
diclofenac
etofenamate
ibuprofen
in vitro permeation test
ketoprofen
naproxen
Journal
Pharmaceutics
ISSN: 1999-4923
Titre abrégé: Pharmaceutics
Pays: Switzerland
ID NLM: 101534003
Informations de publication
Date de publication:
20 Aug 2021
20 Aug 2021
Historique:
received:
30
06
2021
revised:
12
08
2021
accepted:
17
08
2021
entrez:
28
8
2021
pubmed:
29
8
2021
medline:
29
8
2021
Statut:
epublish
Résumé
Pharmaceutical products containing non-steroidal anti-inflammatory drugs (NSAIDs) are among the most prescribed topical formulations used for analgesic and antirheumatic properties. These drugs must overcome the skin barrier to cause a therapeutic effect. Human skin has been widely used as a model to study in vitro drug diffusion and permeation, however, it suffers from many limitations. Therefore, to perform in vitro permeation test (IVPT), we used a Strat-M
Identifiants
pubmed: 34452264
pii: pharmaceutics13081305
doi: 10.3390/pharmaceutics13081305
pmc: PMC8398299
pii:
doi:
Types de publication
Journal Article
Langues
eng
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