Drug Release and Pharmacokinetic Evaluation of Novel Implantable Mometasone Furoate Matrices in Rabbit Maxillary Sinuses.

bioresorbable chronic rhinosinusitis corticosteroid drug delivery drug matrix mometasone furoate mucosa nasal implant pharmacokinetics sustained release

Journal

American journal of rhinology & allergy
ISSN: 1945-8932
Titre abrégé: Am J Rhinol Allergy
Pays: United States
ID NLM: 101490775

Informations de publication

Date de publication:
Mar 2022
Historique:
pubmed: 1 9 2021
medline: 4 2 2022
entrez: 31 8 2021
Statut: ppublish

Résumé

Intranasal corticosteroid sprays (INCSs) used to treat chronic rhinosinusitis are suboptimal due to limited penetration into the middle meatus, rapid clearance, and poor patient compliance. A bioresorbable drug matrix, developed with the XTreo To evaluate the in vitro drug release and in vivo pharmacokinetics of novel mometasone furoate (MF) matrices in a rabbit dorsal maxillary osteotomy model. XTreo XTreo The XTreo

Sections du résumé

BACKGROUND BACKGROUND
Intranasal corticosteroid sprays (INCSs) used to treat chronic rhinosinusitis are suboptimal due to limited penetration into the middle meatus, rapid clearance, and poor patient compliance. A bioresorbable drug matrix, developed with the XTreo
OBJECTIVE OBJECTIVE
To evaluate the in vitro drug release and in vivo pharmacokinetics of novel mometasone furoate (MF) matrices in a rabbit dorsal maxillary osteotomy model.
METHODS METHODS
XTreo
RESULTS RESULTS
XTreo
CONCLUSION CONCLUSIONS
The XTreo

Identifiants

pubmed: 34463546
doi: 10.1177/19458924211039197
doi:

Substances chimiques

Nasal Sprays 0
Mometasone Furoate 04201GDN4R

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

198-206

Auteurs

Changcheng You (C)

Lyra Therapeutics, Inc., Watertown, Massachusetts.

Ling-Fang Tseng (LF)

Lyra Therapeutics, Inc., Watertown, Massachusetts.

Alexander Pappas (A)

Lyra Therapeutics, Inc., Watertown, Massachusetts.

Danny Concagh (D)

Lyra Therapeutics, Inc., Watertown, Massachusetts.

Yina Kuang (Y)

Lyra Therapeutics, Inc., Watertown, Massachusetts.

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Classifications MeSH