Untangling the web of 5-lipoxygenase-derived products from a molecular and structural perspective: The battle between pro- and anti-inflammatory lipid mediators.


Journal

Biochemical pharmacology
ISSN: 1873-2968
Titre abrégé: Biochem Pharmacol
Pays: England
ID NLM: 0101032

Informations de publication

Date de publication:
11 2021
Historique:
received: 12 07 2021
revised: 29 08 2021
accepted: 01 09 2021
pubmed: 7 9 2021
medline: 7 1 2022
entrez: 6 9 2021
Statut: ppublish

Résumé

Arachidonic acid (AA) is the precursor to leukotrienes (LT), potent mediators of the inflammatory response. In the 35 + years since cysteinyl-LTs were reported to mediate antigen-induced constriction of bronchi in tissue from asthma patients, numerous cellular responses evoked by the LTs, such as chemoattraction and G protein-coupled receptor (GPCR) activation, have been elucidated and revealed a potential for 5-lipoxygenase (5-LOX) as a promising drug target that goes beyond asthma. We describe herein early work identifying 5-LOX as the key enzyme that initiates LT biosynthesis and the discovery of its membrane-embedded helper protein required to execute the two-step reaction that transforms AA to the progenitor leukotriene A

Identifiants

pubmed: 34487716
pii: S0006-2952(21)00375-0
doi: 10.1016/j.bcp.2021.114759
pmc: PMC8865081
mid: NIHMS1740068
pii:
doi:

Substances chimiques

Anti-Inflammatory Agents 0
Lipids 0
Arachidonate 5-Lipoxygenase EC 1.13.11.34

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

114759

Subventions

Organisme : NHLBI NIH HHS
ID : R01 HL107887
Pays : United States
Organisme : NIGMS NIH HHS
ID : R15 GM143724
Pays : United States

Informations de copyright

Copyright © 2021. Published by Elsevier Inc.

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Auteurs

Nathaniel C Gilbert (NC)

Department of Biological Sciences, Louisiana State University, Baton Rouge, LA, USA. Electronic address: ngilbert@lsu.edu.

Marcia E Newcomer (ME)

Department of Biological Sciences, Louisiana State University, Baton Rouge, LA, USA.

Oliver Werz (O)

Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, Friedrich-Schiller-University Jena, 07743 Jena, Germany.

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Classifications MeSH