Xanthopsin-Like Systems via Site-Specific Click-Functionalization of a Retinoic Acid Binding Protein.

Morita-Baylis-Hillman adducts PYP-like chromophores light-sensitive proteins site-specific reactions synthetic xanthopsin-like proteins

Journal

Chembiochem : a European journal of chemical biology
ISSN: 1439-7633
Titre abrégé: Chembiochem
Pays: Germany
ID NLM: 100937360

Informations de publication

Date de publication:
05 01 2022
Historique:
revised: 12 10 2021
received: 25 08 2021
pubmed: 15 10 2021
medline: 22 2 2022
entrez: 14 10 2021
Statut: ppublish

Résumé

The use of light-responsive proteins to control both living or synthetic cells, is at the core of the expanding fields of optogenetics and synthetic biology. It is thus apparent that a richer reaction toolbox for the preparation of such systems is of fundamental importance. Here, we provide a proof-of-principle demonstration that Morita-Baylis-Hillman adducts can be employed to perform a facile site-specific, irreversible and diastereoselective click-functionalization of a lysine residue buried into a lipophilic binding pocket and yielding an unnatural chromophore with an extended π-system. In doing so we effectively open the path to the in vitro preparation of a library of synthetic proteins structurally reminiscent of xanthopsin eubacterial photoreceptors. We argue that such a library, made of variable unnatural chromophores inserted in an easy-to-mutate and crystallize retinoic acid transporter, significantly expand the scope of the recently introduced rhodopsin mimics as both optogenetic and "lab-on-a-molecule" tools.

Identifiants

pubmed: 34647400
doi: 10.1002/cbic.202100449
pmc: PMC8934143
mid: NIHMS1775712
doi:

Substances chimiques

Receptors, Retinoic Acid 0
Rhodopsin 9009-81-8

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

e202100449

Subventions

Organisme : NIGMS NIH HHS
ID : R15 GM126627
Pays : United States
Organisme : Italian MIUR
ID : PRIN 2015

Informations de copyright

© 2021 Wiley-VCH GmbH.

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Auteurs

Giusy Tassone (G)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Marco Paolino (M)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Cecilia Pozzi (C)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Annalisa Reale (A)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Laura Salvini (L)

Toscana Life Sciences Foundation, Via Fiorentina 1, 53100, Siena, Italy.

Gianluca Giorgi (G)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Maurizio Orlandini (M)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Federico Galvagni (F)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Stefano Mangani (S)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

Xuchun Yang (X)

Chemistry Department, Bowling Green State University, Overman Hall, Bowling Green, OH 43403, USA.

Benedetta Carlotti (B)

Dipartimento di Chimica, Biologia e Biotecnologie, Università di Perugia, Via Elce di Sotto, 8, 06123, Perugia, Italy.

Fausto Ortica (F)

Dipartimento di Chimica, Biologia e Biotecnologie, Università di Perugia, Via Elce di Sotto, 8, 06123, Perugia, Italy.

Loredana Latterini (L)

Dipartimento di Chimica, Biologia e Biotecnologie, Università di Perugia, Via Elce di Sotto, 8, 06123, Perugia, Italy.

Massimo Olivucci (M)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.
Chemistry Department, Bowling Green State University, Overman Hall, Bowling Green, OH 43403, USA.

Andrea Cappelli (A)

Dipartimento di Biotecnologie, Chimica e Farmacia, Dipartimento di Eccellenza 2018-2022), Università degli Studi di Siena, Via A. Moro 2, 53100, Siena, Italy.

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