A Novel Antagonist Peptide Reveals a Physiological Role of Insulin-Like Peptide 5 in Control of Colorectal Function.
Journal
ACS pharmacology & translational science
ISSN: 2575-9108
Titre abrégé: ACS Pharmacol Transl Sci
Pays: United States
ID NLM: 101721411
Informations de publication
Date de publication:
08 Oct 2021
08 Oct 2021
Historique:
received:
06
07
2021
entrez:
18
10
2021
pubmed:
19
10
2021
medline:
19
10
2021
Statut:
epublish
Résumé
Insulin-like peptide 5 (INSL5), the natural ligand for the relaxin family peptide receptor 4 (RXFP4), is a gut hormone that is exclusively produced by colonic L-cells. We have recently developed an analogue of INSL5, INSL5-A13, that acts as an RXFP4 agonist
Identifiants
pubmed: 34661082
doi: 10.1021/acsptsci.1c00171
pmc: PMC8506612
doi:
Types de publication
Journal Article
Langues
eng
Pagination
1665-1674Informations de copyright
© 2021 American Chemical Society.
Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
Références
J Am Chem Soc. 2011 Apr 6;133(13):4965-74
pubmed: 21384867
FASEB J. 2007 Mar;21(3):754-65
pubmed: 17197386
J Mol Endocrinol. 2018 Apr;60(3):213-224
pubmed: 29535183
J Biomol Screen. 2008 Oct;13(9):888-98
pubmed: 18812574
J Biol Chem. 2006 May 12;281(19):13068-13074
pubmed: 16547350
Proc Natl Acad Sci U S A. 2014 Jul 29;111(30):11133-8
pubmed: 25028498
J Biol Chem. 2007 Aug 31;282(35):25425-35
pubmed: 17606621
Mol Metab. 2018 May;11:70-83
pubmed: 29576437
Biopolymers. 2011;96(1):81-7
pubmed: 20560146
J Med Chem. 2013 Dec 12;56(23):9509-16
pubmed: 24188028
Genomics. 1999 Aug 15;60(1):50-6
pubmed: 10458910
Cell Metab. 2017 Apr 4;25(4):777-796
pubmed: 28380372
Lancet. 2012 Jun 9;379(9832):2151-61
pubmed: 22579125
Bioconjug Chem. 2008 Jul;19(7):1456-63
pubmed: 18529069
Cell Tissue Res. 2006 Jun;324(3):353-60
pubmed: 16453106
Prog Neurobiol. 2004 Feb;72(2):143-64
pubmed: 15063530
JAMA. 2019 Mar 5;321(9):891-892
pubmed: 30763429
Neuroscience. 2000;101(2):459-69
pubmed: 11074168
Sci Rep. 2019 Nov 28;9(1):17828
pubmed: 31780677
ACS Chem Neurosci. 2020 Jul 15;11(14):2077-2084
pubmed: 32519845
Arch Biochem Biophys. 2017 Apr 1;619:27-34
pubmed: 28274616
Br J Pharmacol. 2017 May;174(10):1077-1089
pubmed: 27243554
Am J Physiol Regul Integr Comp Physiol. 2003 May;284(5):R1269-76
pubmed: 12676748
Amino Acids. 2016 Apr;48(4):987-992
pubmed: 26661035
Neurogastroenterol Motil. 2005 Aug;17(4):585-94
pubmed: 16078948
Arch Biochem Biophys. 2014 Sep 15;558:127-32
pubmed: 25043977
J Biol Chem. 2008 Aug 29;283(35):23811-8
pubmed: 18577524
J Med Chem. 2016 Mar 10;59(5):2118-25
pubmed: 26824523
Am J Physiol. 1998 Dec;275(6):G1415-22
pubmed: 9843779
Naunyn Schmiedebergs Arch Pharmacol. 2017 Jan;390(1):105-111
pubmed: 27888281
J Physiol. 1985 Nov;368:667-78
pubmed: 2867220
Mol Metab. 2018 Oct;16:65-75
pubmed: 30104166
Diabetologia. 2020 Jul;63(7):1396-1407
pubmed: 32342115
Neurogastroenterol Motil. 2020 May;32(5):e13796
pubmed: 31989750
Amino Acids. 2010 Jul;39(2):409-16
pubmed: 20043231
Mol Metab. 2019 Nov;29:158-169
pubmed: 31668387
J Biol Chem. 2005 Jan 7;280(1):292-300
pubmed: 15525639
Chembiochem. 2008 Jul 21;9(11):1816-22
pubmed: 18576448