Pharmacokinetics of cannabichromene in a medical cannabis product also containing cannabidiol and Δ


Journal

European journal of clinical pharmacology
ISSN: 1432-1041
Titre abrégé: Eur J Clin Pharmacol
Pays: Germany
ID NLM: 1256165

Informations de publication

Date de publication:
Feb 2022
Historique:
received: 28 04 2021
accepted: 11 10 2021
pubmed: 20 10 2021
medline: 26 2 2022
entrez: 19 10 2021
Statut: ppublish

Résumé

Cannabichromene (CBC) is a phytocannabinoid commonly found in cannabis, yet its acute post-dose pharmacokinetics (PK) have not been examined in humans. This is a secondary data analysis from a trial investigating Spectrum Yellow oil, an oral cannabis product used for medical purposes that contained 20 mg cannabidiol (CBD), 0.9 mg Δ Participants (N = 43) were randomized to one of 5 groups: 120 mg CBD, 5.4 mg THC, and 6.6 mg CBC daily; 240 mg CBD, 10.8 mg THC, and 13.2 mg CBC daily; 360 mg CBD, 16.2 mg THC, and 19.8 mg CBC daily; 480 mg CBD, 21.6 mg THC, and 26.4 mg CBC daily; or placebo. Study medication was administered every 12 h for 7 days. Plasma CBC concentrations were analyzed by a validated two-dimensional high-performance liquid chromatography-tandem mass spectrometry assay. After a single dose and after the final dose, the C CBC may have preferential absorption over CBD and THC when administered together. Australian New Zealand Clinical Trials Registry #ACTRN12619001450101, registered 18 October 2019.

Identifiants

pubmed: 34664109
doi: 10.1007/s00228-021-03232-8
pii: 10.1007/s00228-021-03232-8
pmc: PMC8748343
doi:

Substances chimiques

Cannabinoids 0
Medical Marijuana 0
Cannabidiol 19GBJ60SN5
Dronabinol 7J8897W37S
cannabichromene K4497H250W

Types de publication

Clinical Trial, Phase I Journal Article Randomized Controlled Trial

Langues

eng

Sous-ensembles de citation

IM

Pagination

259-265

Informations de copyright

© 2021. The Author(s).

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Auteurs

Erica N Peters (EN)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada. erica.peters@canopygrowth.com.

Laura MacNair (L)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

Irina Mosesova (I)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

Uwe Christians (U)

iC42 Clinical Research and Development, Department of Anesthesiology, University of Colorado Anschutz Medical Campus, Aurora, CO, USA.

Cristina Sempio (C)

iC42 Clinical Research and Development, Department of Anesthesiology, University of Colorado Anschutz Medical Campus, Aurora, CO, USA.

Jost Klawitter (J)

iC42 Clinical Research and Development, Department of Anesthesiology, University of Colorado Anschutz Medical Campus, Aurora, CO, USA.

M Hunter Land (MH)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

Mark A Ware (MA)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

Cynthia Turcotte (C)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

Marcel O Bonn-Miller (MO)

Canopy Growth Corporation, One Hershey Drive, Smiths Falls, ON, Canada.

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Classifications MeSH