Formulation and In-Vitro Characterization of pH-Responsive Semi-Interpenetrating Polymer Network Hydrogels for Controlled Release of Ketorolac Tromethamine.

carbopol 934 hydrogel ketorolac tromethamine sodium polystyrene sulfonate

Journal

Gels (Basel, Switzerland)
ISSN: 2310-2861
Titre abrégé: Gels
Pays: Switzerland
ID NLM: 101696925

Informations de publication

Date de publication:
13 Oct 2021
Historique:
received: 06 09 2021
revised: 06 10 2021
accepted: 09 10 2021
entrez: 26 10 2021
pubmed: 27 10 2021
medline: 27 10 2021
Statut: epublish

Résumé

Ketorolac tromethamine is a non-steroidal anti-inflammatory drug used in the management of severe pain. The half-life of Ketorolac tromethamine is within the range of 2.5-4 h. Hence, repeated doses of Ketorolac tromethamine are needed in a day to maintain the therapeutic level. However, taking several doses of Ketorolac tromethamine in a day generates certain complications, such as acute renal failure and gastrointestinal ulceration. Therefore, a polymeric-controlled drug delivery system is needed that could prolong the release of Ketorolac tromethamine. Therefore, in the current study, pH-responsive carbopol 934/sodium polystyrene sulfonate-co-poly(acrylic acid) (CP/SpScPAA) hydrogels were developed by the free radical polymerization technique for the controlled release of Ketorolac tromethamine. Monomer acrylic acid was crosslinked with the polymers carbopol 934 and sodium polystyrene sulfonate by the cross-linker

Identifiants

pubmed: 34698162
pii: gels7040167
doi: 10.3390/gels7040167
pmc: PMC8544598
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : National Science Council of Taiwan
ID : MOST 110-2320-B-037-014-MY2
Organisme : Kaohsiung Medical University Research Foundation
ID : KMU-TC109A03-1

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Auteurs

Muhammad Suhail (M)

School of Pharmacy, Kaohsiung Medical University, Kaohsiung City 80708, Taiwan.

Yi-Han Hsieh (YH)

Department of Biomedical Science and Environmental Biology, Kaohsiung Medical University, Kaohsiung City 80708, Taiwan.

Yu-Fang Shao (YF)

Department of Biomedical Science and Environmental Biology, Kaohsiung Medical University, Kaohsiung City 80708, Taiwan.

Muhammad Usman Minhas (MU)

College of Pharmacy, University of Sargodha, Sargodha 40100, Pakistan.

Pao-Chu Wu (PC)

School of Pharmacy, Kaohsiung Medical University, Kaohsiung City 80708, Taiwan.
Department of Medical Research, Kaohsiung Medical University Hospital, Kaohsiung 80708, Taiwan.
Drug Development and Value Creation Research Center, Kaohsiung Medical University, Kaohsiung 80708, Taiwan.

Classifications MeSH