Machine Learning Models for Human

clinical data compound design human pharmacokinetics machine learning pharmacokinetic modeling structure−property relationships

Journal

Molecular pharmaceutics
ISSN: 1543-8392
Titre abrégé: Mol Pharm
Pays: United States
ID NLM: 101197791

Informations de publication

Date de publication:
06 12 2021
Historique:
pubmed: 12 11 2021
medline: 15 3 2022
entrez: 11 11 2021
Statut: ppublish

Résumé

Prior to clinical development, a comprehensive pharmacokinetic characterization of a novel drug is required to understand its exposure at the site of action and elimination. Accordingly,

Identifiants

pubmed: 34758626
doi: 10.1021/acs.molpharmaceut.1c00718
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

4520-4530

Auteurs

Filip Miljković (F)

Data Science and AI, Imaging and Data Analytics, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Gothenburg SE-43183, Sweden.

Anton Martinsson (A)

Data Science and AI, Imaging and Data Analytics, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Gothenburg SE-43183, Sweden.

Olga Obrezanova (O)

Data Science and AI, Imaging and Data Analytics, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Cambridge CB4 0FZ, U.K.

Beth Williamson (B)

Drug Metabolism and Pharmacokinetics, Research and Early Development, Oncology, R&D, AstraZeneca, Cambridge CB10 1XL, U.K.

Martin Johnson (M)

Clinical Pharmacology & Quantitative Pharmacology, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Cambridge SG8 6HB, U.K.

Andy Sykes (A)

Clinical Pharmacology & Quantitative Pharmacology, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Cambridge SG8 6HB, U.K.

Andreas Bender (A)

Data Science and AI, Imaging and Data Analytics, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Cambridge CB4 0FZ, U.K.
Department of Chemistry, Centre for Molecular Informatics, University of Cambridge, Cambridge CB2 1EW, U.K.

Nigel Greene (N)

Data Science and AI, Imaging and Data Analytics, Clinical Pharmacology & Safety Sciences, R&D, AstraZeneca, Waltham, Massachusetts 02451, United States.

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Classifications MeSH