Phthalimide analogs for antimalarial drug discovery.
Journal
RSC medicinal chemistry
ISSN: 2632-8682
Titre abrégé: RSC Med Chem
Pays: England
ID NLM: 101759460
Informations de publication
Date de publication:
17 Nov 2021
17 Nov 2021
Historique:
received:
20
07
2021
accepted:
03
08
2021
entrez:
26
11
2021
pubmed:
27
11
2021
medline:
27
11
2021
Statut:
epublish
Résumé
Malaria remains one of the world's most life-threatening diseases and, thus, it is a major public health concern all around the world. The disease can become devastating if not treated with proper medication in a timely manner. Currently, the number of viable treatment therapies is in continuous decline due to compromised effectiveness, probably owing to the complex life cycle of
Identifiants
pubmed: 34825184
doi: 10.1039/d1md00244a
pii: d1md00244a
pmc: PMC8597421
doi:
Types de publication
Journal Article
Review
Langues
eng
Pagination
1854-1867Informations de copyright
This journal is © The Royal Society of Chemistry.
Déclaration de conflit d'intérêts
We declare no conflicts of interest.
Références
Nat Chem Biol. 2019 Nov;15(11):1077-1084
pubmed: 31591562
Med Res Rev. 2018 Sep;38(5):1511-1535
pubmed: 29372568
Phytother Res. 2008 Dec;22(12):1570-6
pubmed: 19067375
PLoS One. 2010 Oct 04;5(10):
pubmed: 20957228
Eur J Med Chem. 2016 Feb 15;109:187-98
pubmed: 26774925
Bioorg Med Chem. 2018 Jul 30;26(13):3837-3844
pubmed: 29983285
Exp Parasitol. 2011 Jun;128(2):97-103
pubmed: 21354139
ACS Omega. 2018 Aug 20;3(8):9424-9430
pubmed: 31459076
Lancet. 1965 Oct 2;2(7414):657-60
pubmed: 4158213
Bioorg Med Chem Lett. 2013 Feb 1;23(3):658-62
pubmed: 23260352
Eur J Med Chem. 2017 Mar 31;129:175-185
pubmed: 28222317
ACS Infect Dis. 2019 Feb 8;5(2):184-198
pubmed: 30554511
Expert Rev Vaccines. 2019 Feb;18(2):133-151
pubmed: 30601095
Mol Microbiol. 2005 Jul;57(2):405-19
pubmed: 15978074
Am J Cancer Res. 2018 Sep 01;8(9):1697-1711
pubmed: 30323964
PLoS One. 2015 Oct 26;10(10):e0139347
pubmed: 26502278
Med Chem. 2012 Mar;8(2):266-72
pubmed: 22385178
Drug Saf Case Rep. 2017 Dec;4(1):6
pubmed: 28258476
ACS Med Chem Lett. 2019 May 23;10(6):887-892
pubmed: 31223443
Am J Trop Med Hyg. 2009 Sep;81(3):525-8
pubmed: 19706926
Malar J. 2016 May 12;15(1):277
pubmed: 27176722
Nature. 2002 Oct 3;419(6906):520-6
pubmed: 12368866
Pharmacol Ther. 2020 Dec;216:107672
pubmed: 32910933
Nat Commun. 2015 Jul 24;6:7690
pubmed: 26205537
Bioorg Med Chem. 2015 Apr 15;23(8):1817-27
pubmed: 25766631
PLoS One. 2016 Mar 02;11(3):e0149996
pubmed: 26934697
Ecancermedicalscience. 2017 Nov 23;11:781
pubmed: 29225688
Bioorg Med Chem. 2021 Jun 1;39:116159
pubmed: 33895706
Malar J. 2014 Aug 30;13:339
pubmed: 25176157
J Med Chem. 2021 Jun 24;64(12):8666-8683
pubmed: 34124905
Acta Trop. 2005 May;94(2):128-38
pubmed: 15817259
J Med Chem. 2011 Jul 14;54(13):4581-9
pubmed: 21644541
Cell Host Microbe. 2019 Jul 10;26(1):35-47
pubmed: 31295423
Antimicrob Agents Chemother. 2015 Jan;59(1):654-8
pubmed: 25313210
ACS Med Chem Lett. 2018 Oct 19;9(12):1205-1210
pubmed: 30613327
Eur J Med Chem. 2010 May;45(5):1731-8
pubmed: 20117861
Int J Parasitol. 2010 Aug 15;40(10):1127-35
pubmed: 20478310
Malar J. 2019 Apr 23;18(1):144
pubmed: 31014336
Blood Cancer J. 2019 Oct 8;9(10):83
pubmed: 31594919
Eur J Med Chem. 2016 Jan 27;108:79-88
pubmed: 26638041
Expert Opin Drug Discov. 2020 Jun;15(6):705-718
pubmed: 32202162
J Med Chem. 2010 Feb 25;53(4):1788-98
pubmed: 20128602
Eur J Med Chem. 2009 Nov;44(11):4778-82
pubmed: 19747753
Curr Med Chem. 2019;26(23):4323-4354
pubmed: 29065822
Bioorg Med Chem Lett. 2020 Jan 15;30(2):126810
pubmed: 31740250
Proc Natl Acad Sci U S A. 2004 Mar 30;101(13):4384-9
pubmed: 15070727
Malar J. 2016 May 20;15(1):284
pubmed: 27206924
Curr Opin Chem Biol. 2019 Oct;52:1-8
pubmed: 30682725
Nat Commun. 2019 Feb 20;10(1):856
pubmed: 30787300
Ann N Y Acad Sci. 2010 Jul;1201:96-103
pubmed: 20649545
Planta Med. 2013 Jan;79(2):150-6
pubmed: 23299758
Bioorg Chem. 2020 Mar;96:103567
pubmed: 32062063
ACS Infect Dis. 2020 Apr 10;6(4):613-628
pubmed: 32078764
Curr Biol. 2019 Jul 8;29(13):R632-R634
pubmed: 31287981
Pharmaceuticals (Basel). 2020 Feb 03;13(2):
pubmed: 32028743
Sci Rep. 2019 Sep 11;9(1):13131
pubmed: 31511546
Bioorg Med Chem Lett. 2012 Apr 15;22(8):2976-9
pubmed: 22414614
Eur J Med Chem. 2018 Jan 1;143:150-156
pubmed: 29174811
Bioorg Med Chem Lett. 2014 Nov 15;24(22):5234-7
pubmed: 25316317
J Chem Inf Model. 2020 Dec 28;60(12):5754-5770
pubmed: 32551639
Pharmacol Ther. 2019 Oct;202:132-139
pubmed: 31202702
Sci Rep. 2017 Jul 27;7(1):6724
pubmed: 28751747
Nat Rev Microbiol. 2009 Dec;7(12):864-74
pubmed: 19881520