Hindrance of the Proteolytic Activity of Neutrophil-Derived Serine Proteases by Serine Protease Inhibitors as a Management of Cardiovascular Diseases and Chronic Inflammation.
COVID-19
SARS-CoV-2
cathepsin G
neutrophil elastase
proteinase 3
serine protease inhibitors
serine proteases
thrombosis
Journal
Frontiers in chemistry
ISSN: 2296-2646
Titre abrégé: Front Chem
Pays: Switzerland
ID NLM: 101627988
Informations de publication
Date de publication:
2021
2021
Historique:
received:
27
09
2021
accepted:
20
10
2021
entrez:
6
12
2021
pubmed:
7
12
2021
medline:
7
12
2021
Statut:
epublish
Résumé
During inflammation neutrophils become activated and segregate neutrophil serine proteases (NSPs) to the surrounding environment in order to support a natural immune defense. However, an excess of proteolytic activity of NSPs can cause many complications, such as cardiovascular diseases and chronic inflammatory disorders, which will be elucidated on a biochemical and immunological level. The application of selective serine protease inhibitors is the logical consequence in the management of the indicated comorbidities and will be summarized in this briefing.
Identifiants
pubmed: 34869231
doi: 10.3389/fchem.2021.784003
pii: 784003
pmc: PMC8634265
doi:
Types de publication
Journal Article
Review
Langues
eng
Pagination
784003Informations de copyright
Copyright © 2021 Burster, Mustafa, Myrzakhmetova, Zhanapiya and Zimecki.
Déclaration de conflit d'intérêts
The authors declare that the research was conducted in the absence of any commercial or financial relationships that could be construed as a potential conflict of interest.
Références
Thromb Haemost. 2010 Sep;104(3):514-22
pubmed: 20589323
J Med Chem. 2017 Jan 26;60(2):658-667
pubmed: 28045523
Mol Med. 2019 May 2;25(1):16
pubmed: 31046673
Nature. 2021 Jul;595(7869):640-644
pubmed: 34321669
Arterioscler Thromb Vasc Biol. 2018 Aug;38(8):1901-1912
pubmed: 29976772
J Clin Med. 2018 Aug 28;7(9):
pubmed: 30154365
Haematologica. 2011 Jul;96(7):954-62
pubmed: 21546506
EBioMedicine. 2016 Aug;10:204-15
pubmed: 27453322
Arch Immunol Ther Exp (Warsz). 2020 Aug 19;68(4):23
pubmed: 32815054
Arch Immunol Ther Exp (Warsz). 1999;47(4):257-64
pubmed: 10483875
Clin Exp Immunol. 2020 Jan;199(1):1-8
pubmed: 31661552
J Biol Chem. 1991 May 25;266(15):9540-8
pubmed: 2033050
Br Heart J. 1993 Apr;69(4):338-42
pubmed: 8489866
Allergy. 2021 Jun;76(6):1846-1858
pubmed: 33484168
Diabetologia. 2019 Dec;62(12):2365-2374
pubmed: 31612267
Antiviral Res. 2013 Dec;100(3):605-14
pubmed: 24121034
Nat Med. 2010 Aug;16(8):887-96
pubmed: 20676107
J Immunol. 2009 Sep 1;183(5):3433-42
pubmed: 19648270
Rev Med Virol. 2021 Mar;31(2):e2157
pubmed: 32844538
FASEB J. 2001 Sep;15(11):2027-9
pubmed: 11511513
Front Immunol. 2017 Nov 06;8:1438
pubmed: 29163511
J Virol. 2000 Aug;74(15):6849-55
pubmed: 10888624
Biochem Biophys Res Commun. 2018 Sep 10;503(3):1284-1290
pubmed: 30017196
Acute Med Surg. 2019 Dec 06;7(1):e471
pubmed: 31988783
J Inflamm Res. 2018 Mar 26;11:123-134
pubmed: 29618937
Biochim Biophys Acta. 1995 Jan 18;1243(1):25-32
pubmed: 7827104
SN Compr Clin Med. 2020;2(8):1103-1108
pubmed: 32838164
Semin Cancer Biol. 2022 May;80:39-57
pubmed: 32027979
Mol Cell. 2020 May 21;78(4):779-784.e5
pubmed: 32362314
J Immunol. 2010 Nov 1;185(9):5360-8
pubmed: 20889553
N Engl J Med. 2020 Feb 20;382(8):727-733
pubmed: 31978945
J Surg Res. 2007 Jun 15;140(2):199-203
pubmed: 17418861
Cell Physiol Biochem. 2019;53(6):982-998
pubmed: 31829530
PLoS One. 2013 Aug 05;8(8):e71447
pubmed: 23940756
Thromb Res. 2020 Nov;195:226-227
pubmed: 32795720
J Thromb Haemost. 2020 May;18(5):1020-1022
pubmed: 32239799
Shock. 2020 Sep;54(3):386-393
pubmed: 31764619
Circulation. 1989 Mar;79(3):549-56
pubmed: 2537159
Biochimie. 2019 Nov;166:142-149
pubmed: 30876969
J Biol Chem. 2015 Oct 2;290(40):24067-78
pubmed: 26269588
Clin Exp Immunol. 2002 Oct;130(1):25-31
pubmed: 12296849
Open Forum Infect Dis. 2020 Nov 19;7(12):ofaa563
pubmed: 33365358
PLoS One. 2016 Mar 17;11(3):e0151509
pubmed: 26986619
Acta Pharmacol Sin. 2020 Sep;41(9):1141-1149
pubmed: 32747721
Nat Rev Nephrol. 2020 Jun;16(6):305-307
pubmed: 32246101
J Virol. 2016 May 27;90(12):5586-5600
pubmed: 27030273
Lancet. 2020 Mar 28;395(10229):1054-1062
pubmed: 32171076
Pulm Pharmacol Ther. 2012 Feb;25(1):99-103
pubmed: 22210005
Structure. 2014 Sep 2;22(9):1333-1340
pubmed: 25156428
Herz. 2020 Jun;45(4):323-324
pubmed: 32274522
J Leukoc Biol. 2017 Sep;102(3):689-698
pubmed: 28546501
Ann Thorac Cardiovasc Surg. 2018 Feb 20;24(1):32-39
pubmed: 29118307
Elife. 2022 Mar 23;11:
pubmed: 35294338
Clin Appl Thromb Hemost. 2008 Apr;14(2):186-92
pubmed: 18372277
Biol Pharm Bull. 2008 Apr;31(4):569-73
pubmed: 18379042
Biochim Biophys Acta Biomembr. 2019 Aug 1;1861(8):1502-1509
pubmed: 31229588
IUBMB Life. 2009 May;61(5):510-5
pubmed: 19180666
J Biol Chem. 2000 Mar 10;275(10):6819-23
pubmed: 10702240
J Am Soc Nephrol. 2002 Dec;13(12):2840-9
pubmed: 12444202
J Thorac Dis. 2014 Dec;6(12):1681-9
pubmed: 25589960
Biochem Biophys Res Commun. 2017 Apr 22;486(1):205-209
pubmed: 28300553
J Immunol. 2014 Feb 15;192(4):1787-95
pubmed: 24446515
Elife. 2020 Jul 07;9:
pubmed: 32633718
Thromb Res. 2020 Oct;194:216-219
pubmed: 33074107
Gastroenterology. 1989 Mar;96(3):853-9
pubmed: 2464526
J Cyst Fibros. 2021 Jan;20(1):31-35
pubmed: 33288475
J Clin Invest. 1994 Sep;94(3):1163-71
pubmed: 8083356
Int Immunopharmacol. 2021 Jun;95:107571
pubmed: 33765614
J Virol. 2013 Jun;87(11):6150-60
pubmed: 23536651
Proc Natl Acad Sci U S A. 2009 Apr 7;106(14):5871-6
pubmed: 19321428
PLoS One. 2020 Oct 20;15(10):e0240012
pubmed: 33079950
Thromb Res. 2010 Aug;126(2):e94-101
pubmed: 20627279
Science. 2020 May 8;368(6491):630-633
pubmed: 32245784
Biochim Biophys Acta. 2000 Jul 14;1480(1-2):245-57
pubmed: 10899625
Respir Res. 2019 Jul 30;20(1):170
pubmed: 31362723
Cells. 2020 Oct 30;9(11):
pubmed: 33143316
J Biol Chem. 1982 Dec 25;257(24):15042-6
pubmed: 6294088
ChemMedChem. 2015 Jul;10(7):1163-73
pubmed: 26083237
Sci Rep. 2018 May 18;8(1):7834
pubmed: 29777136
J Immunol. 2017 Feb 15;198(4):1474-1483
pubmed: 28053237
Front Immunol. 2019 May 09;10:1037
pubmed: 31143182
Int J Mol Sci. 2021 Jan 13;22(2):
pubmed: 33450865
Chest. 2017 Aug;152(2):249-262
pubmed: 28442313
Basic Res Cardiol. 2017 Sep 14;112(6):62
pubmed: 28913553
Biomolecules. 2019 May 29;9(6):
pubmed: 31146486
Inflamm Res. 2009 Apr;58(4):198-203
pubmed: 19169649
Thromb Res. 2021 Jan;197:65-68
pubmed: 33186849
COPD. 2018 Oct;15(5):472-478
pubmed: 30822244
Thromb J. 2019 Mar 29;17:4
pubmed: 30976204
Shock. 2010 Jan;33(1):14-8
pubmed: 19487982
Antioxid Redox Signal. 2016 May 10;24(14):813-36
pubmed: 26981846
Ann Intern Med. 2020 Aug 18;173(4):268-277
pubmed: 32374815
Int J Mol Sci. 2020 Jan 19;21(2):
pubmed: 31963828
Sci Rep. 2016 Apr 22;6:24880
pubmed: 27101808
Am J Respir Crit Care Med. 2010 Feb 1;181(3):247-53
pubmed: 19875688
Can J Physiol Pharmacol. 2002 Apr;80(4):346-53
pubmed: 12025971
Biochem Pharmacol. 2019 Jun;164:349-367
pubmed: 30978322
Cell Mol Immunol. 2020 Jun;17(6):647-649
pubmed: 32313207
Proc Natl Acad Sci U S A. 2006 Feb 28;103(9):3316-21
pubmed: 16488976
Infect Immun. 2000 Dec;68(12):6519-25
pubmed: 11083760
Drugs. 2020 Sep;80(14):1383-1396
pubmed: 32705604
Med Res Rev. 2013 Jun;33 Suppl 1:E73-101
pubmed: 21681767
Cancer Discov. 2020 Jun;10(6):779-782
pubmed: 32276929
J Virol. 2010 Dec;84(24):12658-64
pubmed: 20926566
J Intern Med. 2005 Jun;257(6):540-8
pubmed: 15910558
Brain Behav Immun. 2021 Mar;93:288-298
pubmed: 33401017
J Cell Mol Med. 2020 Oct;24(20):11998-12007
pubmed: 32935466
Clin Chem Lab Med. 2021 Mar 08;59(8):e330-e334
pubmed: 33675194
Biochem Pharmacol. 2006 Jan 12;71(3):287-93
pubmed: 16310171
J Clin Pharm Ther. 2020 Dec;45(6):1515-1519
pubmed: 32860252
EClinicalMedicine. 2021 May;35:100849
pubmed: 33903855
FASEB J. 2014 May;28(5):2318-31
pubmed: 24532668
N Engl J Med. 2013 May 23;368(21):1963-70
pubmed: 23692169
PLoS One. 2018 Apr 13;13(4):e0195077
pubmed: 29652924
Life Sci. 2017 Oct 1;186:118-124
pubmed: 28801264
EBioMedicine. 2020 Sep;59:102969
pubmed: 32853989
Annu Rev Biochem. 1991;60:443-75
pubmed: 1883201
Front Immunol. 2019 Mar 28;10:600
pubmed: 30984180
FEBS Lett. 1996 May 13;386(1):82-6
pubmed: 8635609
Clin Exp Rheumatol. 2008 May-Jun;26(3 Suppl 49):S112-7
pubmed: 18799068
Circulation. 2016 Oct 18;134(16):1176-1188
pubmed: 27660294
Intern Med. 2021 Jan 1;60(1):145-150
pubmed: 32830174
J Cyst Fibros. 2016 May;15(3):325-31
pubmed: 26526358
Curr Pharm Des. 2011 Dec;17(38):4308-17
pubmed: 22204429
Biochem Cell Biol. 2021 Feb;99(1):47-53
pubmed: 32476452
J Intensive Care. 2014 Dec 31;2(1):67
pubmed: 25705423
Proc Natl Acad Sci U S A. 2012 Apr 17;109(16):6229-34
pubmed: 22474388
Int J Biochem Cell Biol. 2008;40(6-7):1317-33
pubmed: 18180196
Br J Pharmacol. 2001 Jun;133(3):422-8
pubmed: 11375259
J Clin Invest. 2014 Oct;124(10):4445-58
pubmed: 25180606
Inflammation. 2012 Feb;35(1):81-8
pubmed: 21246269
Crit Care. 2006;10(6):317
pubmed: 17096866
Arch Immunol Ther Exp (Warsz). 2020 Aug 19;68(4):25
pubmed: 32815043
J Biol Chem. 1994 Nov 25;269(47):29502-8
pubmed: 7961933
Biochimie. 2008 Feb;90(2):227-42
pubmed: 18021746
Emerg Microbes Infect. 2021 Dec;10(1):317-330
pubmed: 33560940
J Cyst Fibros. 2020 Mar;19(2):299-304
pubmed: 31501052
Scand J Rheumatol. 2012 Mar;41(2):116-9
pubmed: 22118245
Anesthesiology. 2015 Oct;123(4):838-50
pubmed: 26270939
J Med Chem. 2020 Nov 25;63(22):13258-13265
pubmed: 32692176
Infect Dis Ther. 2020 Jun;9(2):241-253
pubmed: 32292686
Biochemistry. 2006 Aug 1;45(30):9104-20
pubmed: 16866356
Diabetes Res Clin Pract. 2020 Jun;164:108220
pubmed: 32442557
J Clin Med. 2020 Apr 15;9(4):
pubmed: 32326602
Front Med (Lausanne). 2018 Aug 03;5:217
pubmed: 30131961
Commun Biol. 2020 Nov 19;3(1):687
pubmed: 33214666
Mol Pharmacol. 2000 Oct;58(4):828-36
pubmed: 10999954
J Clin Invest. 1981 Aug;68(2):484-90
pubmed: 7021592
Front Pharmacol. 2020 Dec 11;11:615398
pubmed: 33362565
PLoS One. 2011;6(8):e22815
pubmed: 21850236
Nat Rev Dis Primers. 2019 Mar 14;5(1):18
pubmed: 30872586
Pharmacol Res. 2020 Jul;157:104859
pubmed: 32360480
Nat Commun. 2020 Mar 27;11(1):1620
pubmed: 32221306
JCI Insight. 2020 Jun 4;5(11):
pubmed: 32329756
Pulm Pharmacol Ther. 2019 Jun;56:86-93
pubmed: 30917927
Kidney Blood Press Res. 2020;45(3):357-362
pubmed: 32450560
Front Immunol. 2020 Mar 03;11:411
pubmed: 32194574
Pharmacol Rev. 2010 Dec;62(4):726-59
pubmed: 21079042
Front Pharmacol. 2020 Aug 06;11:1124
pubmed: 32848743
EBioMedicine. 2020 May;55:102763
pubmed: 32361250
J Phys Chem Lett. 2020 Aug 20;11(16):6655-6663
pubmed: 32787225
Am J Pathol. 2014 Aug;184(8):2197-210
pubmed: 24929239
Annu Rev Cell Dev Biol. 2020 Oct 6;36:191-218
pubmed: 32663035
J Immunol. 1998 Feb 1;160(3):1436-43
pubmed: 9570564
Biol Chem. 2005 Aug;386(8):801-11
pubmed: 16201876
PLoS One. 2019 Oct 24;14(10):e0220022
pubmed: 31647805
JAMA. 2007 Feb 7;297(5):471-9
pubmed: 17284697
Thromb Res. 2020 Dec;196:483-485
pubmed: 33091700
Arterioscler Thromb Vasc Biol. 2001 Sep;21(9):1538-43
pubmed: 11557685
EBioMedicine. 2020 Aug;58:102925
pubmed: 32745993
FEBS J. 2020 Sep;287(18):4068-4081
pubmed: 31995266
Clin Pharmacokinet. 2011 Jun;50(6):349-69
pubmed: 21553931
J Biol Chem. 2020 Dec 18;295(51):17624-17631
pubmed: 33454002
Proc Natl Acad Sci U S A. 2014 Oct 21;111(42):15214-9
pubmed: 25288733
ACS Omega. 2021 Mar 05;6(10):7181-7185
pubmed: 33748632
Cell. 2020 Apr 16;181(2):271-280.e8
pubmed: 32142651
Bioorg Med Chem. 2009 May 1;17(9):3302-7
pubmed: 19362846
Int J Mol Sci. 2021 Jul 27;22(15):
pubmed: 34360796
Am J Transl Res. 2017 Nov 15;9(11):5127-5137
pubmed: 29218110
Antimicrob Agents Chemother. 2020 May 21;64(6):
pubmed: 32312781
Microb Pathog. 2020 Dec;149:104504
pubmed: 32950636
Nat Rev Immunol. 2020 Jun;20(6):363-374
pubmed: 32346093
Eur Heart J. 2000 Oct;21(19):1607-13
pubmed: 10988013
Eur J Pharmacol. 1992 Jun 17;216(3):401-5
pubmed: 1425930
Cell Rep. 2019 Jun 18;27(12):3646-3656.e5
pubmed: 31216481
Biochem Biophys Res Commun. 1985 Mar 15;127(2):443-9
pubmed: 3884010
Br Heart J. 1990 Feb;63(2):82-7
pubmed: 2317413
Arch Surg. 1998 Sep;133(9):1002-6
pubmed: 9749856
Expert Opin Ther Pat. 2013 Dec;23(12):1611-24
pubmed: 24079661
Proc Natl Acad Sci U S A. 1998 Oct 13;95(21):12641-6
pubmed: 9770539
Am J Pathol. 2019 Aug;189(8):1526-1535
pubmed: 31108101
PLoS One. 2021 May 26;16(5):e0251426
pubmed: 34038453
Circulation. 1990 Sep;82(3 Suppl):II47-59
pubmed: 2203564
Br J Anaesth. 2002 Jun;88(6):848-63
pubmed: 12173205
J Mol Cell Cardiol. 2019 Sep;134:29-39
pubmed: 31252040
Life Sci Alliance. 2020 Jul 23;3(9):
pubmed: 32703818
Infect Genet Evol. 2021 Jun;90:104760
pubmed: 33556558
N Engl J Med. 2020 Apr 23;382(17):1653-1659
pubmed: 32227760
Clin Appl Thromb Hemost. 2006 Jan;12(1):47-54
pubmed: 16444434
FASEB J. 2019 Jan;33(1):1401-1414
pubmed: 30130433