Safety and efficacy of hydroxychloroquine for treatment of non-severe COVID-19 among adults in Uganda: a randomized open label phase II clinical trial.


Journal

BMC infectious diseases
ISSN: 1471-2334
Titre abrégé: BMC Infect Dis
Pays: England
ID NLM: 100968551

Informations de publication

Date de publication:
06 Dec 2021
Historique:
received: 08 05 2021
accepted: 22 11 2021
entrez: 7 12 2021
pubmed: 8 12 2021
medline: 15 12 2021
Statut: epublish

Résumé

Several repurposed drugs such as hydroxychloroquine (HCQ) have been investigated for treatment of COVID-19, but none was confirmed to be efficacious. While in vitro studies have demonstrated antiviral properties of HCQ, data from clinical trials were conflicting regarding its benefit for COVID-19 treatment. Drugs that limit viral replication may be beneficial in the earlier course of the disease thus slowing progression to severe and critical illness. We conducted a randomized open label Phase II clinical trial from October-December 2020. Patients diagnosed with COVID-19 using RT-PCR were included in the study if they were 18 years and above and had a diagnosis of COVID-19 made in the last 3 days. Patients were randomized in blocks, to receive either HCQ 400 mg twice a day for the first day followed by 200 mg twice daily for the next 4 days plus standard of care (SOC) treatment or SOC treatment alone. SARS COV-2 viral load (CT values) from RT-PCR testing of samples collected using nasal/orapharyngeal swabs was performed at baseline, day 2, 4, 6, 8 and 10. The primary outcome was median time from randomization to SARS COV-2 viral clearance by day 6. Of the 105 participants enrolled, 55 were assigned to the intervention group (HCQ plus SOC) and 50 to the control group (SOC only). Baseline characteristics were similar across treatment arms. Viral clearance did not differ by treatment arm, 20 and 19 participants respectively had SARS COV-2 viral load clearance by day 6 with no significant difference, median (IQR) number of days to viral load clearance between the two groups was 4(3-4) vs 4(2-4): p = 0.457. There were no significant differences in secondary outcomes (symptom resolution and adverse events) between the intervention group and the control group. There were no significant differences in specific adverse events such as elevated alkaline phosphatase, prolonged QTc interval on ECG, among patients in the intervention group as compared to the control group. Our results show that HCQ 400 mg twice a day for the first day followed by 200 mg twice daily for the next 4 days was safe but not associated with reduction in viral clearance or symptom resolution among adults with COVID-19 in Uganda.  NCT04860284.

Sections du résumé

BACKGROUND BACKGROUND
Several repurposed drugs such as hydroxychloroquine (HCQ) have been investigated for treatment of COVID-19, but none was confirmed to be efficacious. While in vitro studies have demonstrated antiviral properties of HCQ, data from clinical trials were conflicting regarding its benefit for COVID-19 treatment. Drugs that limit viral replication may be beneficial in the earlier course of the disease thus slowing progression to severe and critical illness.
DESIGN METHODS
We conducted a randomized open label Phase II clinical trial from October-December 2020.
METHODS METHODS
Patients diagnosed with COVID-19 using RT-PCR were included in the study if they were 18 years and above and had a diagnosis of COVID-19 made in the last 3 days. Patients were randomized in blocks, to receive either HCQ 400 mg twice a day for the first day followed by 200 mg twice daily for the next 4 days plus standard of care (SOC) treatment or SOC treatment alone. SARS COV-2 viral load (CT values) from RT-PCR testing of samples collected using nasal/orapharyngeal swabs was performed at baseline, day 2, 4, 6, 8 and 10. The primary outcome was median time from randomization to SARS COV-2 viral clearance by day 6.
RESULTS RESULTS
Of the 105 participants enrolled, 55 were assigned to the intervention group (HCQ plus SOC) and 50 to the control group (SOC only). Baseline characteristics were similar across treatment arms. Viral clearance did not differ by treatment arm, 20 and 19 participants respectively had SARS COV-2 viral load clearance by day 6 with no significant difference, median (IQR) number of days to viral load clearance between the two groups was 4(3-4) vs 4(2-4): p = 0.457. There were no significant differences in secondary outcomes (symptom resolution and adverse events) between the intervention group and the control group. There were no significant differences in specific adverse events such as elevated alkaline phosphatase, prolonged QTc interval on ECG, among patients in the intervention group as compared to the control group.
CONCLUSION CONCLUSIONS
Our results show that HCQ 400 mg twice a day for the first day followed by 200 mg twice daily for the next 4 days was safe but not associated with reduction in viral clearance or symptom resolution among adults with COVID-19 in Uganda.
TRIAL REGISTRATION BACKGROUND
 NCT04860284.

Identifiants

pubmed: 34872511
doi: 10.1186/s12879-021-06897-9
pii: 10.1186/s12879-021-06897-9
pmc: PMC8647506
doi:

Substances chimiques

Hydroxychloroquine 4QWG6N8QKH

Banques de données

ClinicalTrials.gov
['NCT04860284']

Types de publication

Clinical Trial, Phase II Journal Article Randomized Controlled Trial

Langues

eng

Sous-ensembles de citation

IM

Pagination

1218

Informations de copyright

© 2021. The Author(s).

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Auteurs

Pauline Byakika-Kibwika (P)

Department of Medicine, Makerere University College of Health Sciences, Makerere University, P.O. Box 7072, Kampala, Uganda. pbyakika@gmail.com.

Christine Sekaggya-Wiltshire (C)

Mulago National Referral Hospital, Kampala, Uganda.
Infectious Diseases Institute, Makerere University, Kampala, Uganda.

Jerome Roy Semakula (JR)

Infectious Diseases Institute, Makerere University, Kampala, Uganda.

Jane Nakibuuka (J)

Mulago National Referral Hospital, Kampala, Uganda.

Joseph Musaazi (J)

Infectious Diseases Institute, Makerere University, Kampala, Uganda.

James Kayima (J)

Department of Medicine, Makerere University College of Health Sciences, Makerere University, P.O. Box 7072, Kampala, Uganda.

Cornelius Sendagire (C)

Department of Anesthesia, Makerere University, Kampala, Uganda.

David Meya (D)

Department of Medicine, Makerere University College of Health Sciences, Makerere University, P.O. Box 7072, Kampala, Uganda.

Bruce Kirenga (B)

Department of Medicine, Makerere University College of Health Sciences, Makerere University, P.O. Box 7072, Kampala, Uganda.
Makerere University Lung Institute, Kampala, Uganda.

Sarah Nanzigu (S)

Department of Pharmacology, Makerere University, Kampala, Uganda.

Arthur Kwizera (A)

Department of Anesthesia, Makerere University, Kampala, Uganda.

Fred Nakwagala (F)

Mulago National Referral Hospital, Kampala, Uganda.

Ivan Kisuule (I)

Mulago National Referral Hospital, Kampala, Uganda.

Misaki Wayengera (M)

Department of Microbiology, Makerere University, Kampala, Uganda.

Henry G Mwebesa (HG)

Ministry of Health, Kampala, Uganda.

Moses R Kamya (MR)

Department of Medicine, Makerere University College of Health Sciences, Makerere University, P.O. Box 7072, Kampala, Uganda.

William Bazeyo (W)

School of Public Health, College of Health Sciences, Makerere University, Kampala, Uganda.

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