Drug Discovery for
Mycobacterium tuberculosis
anti-tuberculosis
computational drug design
molecular docking
structure-based drug design
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
09 Dec 2021
09 Dec 2021
Historique:
received:
15
10
2021
revised:
09
11
2021
accepted:
14
11
2021
entrez:
24
12
2021
pubmed:
25
12
2021
medline:
2
2
2022
Statut:
epublish
Résumé
Developing new, more effective antibiotics against resistant
Identifiants
pubmed: 34948055
pii: ijms222413259
doi: 10.3390/ijms222413259
pmc: PMC8703488
pii:
doi:
Substances chimiques
Antitubercular Agents
0
Types de publication
Journal Article
Review
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : National Research Foundation
ID : 110906.
Références
Tuberculosis (Edinb). 2010 Jul;90(4):225-35
pubmed: 20488753
Nat Chem Biol. 2007 Jun;3(6):323-4
pubmed: 17496888
Nucleic Acids Res. 2016 Jan 4;44(D1):D1202-13
pubmed: 26400175
Int J Mycobacteriol. 2014 Dec;3(4):276-82
pubmed: 26786627
PLoS One. 2011;6(12):e28428
pubmed: 22164290
Curr Med Chem. 2006;13(25):2995-3003
pubmed: 17073642
J Clin Microbiol. 2017 Nov;55(11):3267-3282
pubmed: 28904183
Pathog Dis. 2017 Jan 1;75(1):
pubmed: 28087649
J Chem Inf Model. 2012 Nov 26;52(11):2864-75
pubmed: 23088335
J Korean Med Sci. 2020 Nov 02;35(42):e379
pubmed: 33140591
Chem Biol. 2003 Sep;10(9):787-97
pubmed: 14522049
Proteins. 2009;77 Suppl 9:114-22
pubmed: 19768677
J Biomol Struct Dyn. 2020 Dec 31;:1-10
pubmed: 33382017
J Comput Chem. 2005 Dec;26(16):1668-88
pubmed: 16200636
Antimicrob Agents Chemother. 2018 Jul 27;62(8):
pubmed: 29784848
Sci Rep. 2018 Aug 16;8(1):12238
pubmed: 30116003
Molecules. 2015 Jul 22;20(7):13384-421
pubmed: 26205061
Int J Mycobacteriol. 2017 Apr-Jun;6(2):142-148
pubmed: 28559515
Drug Des Devel Ther. 2017 Mar 02;11:563-574
pubmed: 28280303
J R Soc Interface. 2012 Dec 7;9(77):3196-207
pubmed: 22933186
Biochemistry. 2008 Apr 8;47(14):4228-36
pubmed: 18335995
Nat Rev Drug Discov. 2005 Aug;4(8):649-63
pubmed: 16056391
Science. 2008 Aug 8;321(5890):792-4
pubmed: 18687952
Curr Opin Chem Biol. 2008 Jun;12(3):372-8
pubmed: 18331851
Antimicrob Agents Chemother. 2002 Feb;46(2):267-74
pubmed: 11796329
Chem Biol. 2015 Jul 23;22(7):917-27
pubmed: 26097035
Future Med Chem. 2011 Apr;3(6):735-50
pubmed: 21554079
Annu Rev Biophys Biomol Struct. 1998;27:249-84
pubmed: 9646869
J Med Chem. 2016 Oct 13;59(19):9269-9275
pubmed: 27589670
Comb Chem High Throughput Screen. 2012 May 1;15(4):328-37
pubmed: 22221065
ACS Med Chem Lett. 2010 Jul 13;1(8):371-5
pubmed: 24900220
J Mol Graph Model. 2021 Jan;102:107770
pubmed: 33065513
J Phys Chem B. 2016 Aug 25;120(33):8313-20
pubmed: 27082121
Drug Des Devel Ther. 2016 Mar 11;10:1147-57
pubmed: 27042006
Methods Mol Biol. 2016;1425:121-37
pubmed: 27311465
Comput Struct Biotechnol J. 2021 Jun 24;19:3708-3719
pubmed: 34285773
Tuberculosis (Edinb). 2009 Sep;89(5):354-63
pubmed: 19783214
Tuberculosis (Edinb). 2011 Jan;91(1):8-13
pubmed: 20980200
Int J Tuberc Lung Dis. 2012 Jun;16(6):724-32
pubmed: 22613684
Curr Protein Pept Sci. 2007 Aug;8(4):365-75
pubmed: 17696869
J Comput Aided Mol Des. 2008 Mar-Apr;22(3-4):133-9
pubmed: 18338228
Lancet Infect Dis. 2015 Nov;15(11):1357-60
pubmed: 26321650
Biochem J. 2001 Feb 1;353(Pt 3):453-8
pubmed: 11171040
N Engl J Med. 2015 Nov 26;373(22):2149-60
pubmed: 26605929
Biochemistry. 2012 Jun 19;51(24):4868-79
pubmed: 22607697
Expert Opin Drug Discov. 2006 Jul;1(2):103-10
pubmed: 23495794
N Engl J Med. 2015 May 28;372(22):2127-35
pubmed: 26017823
Clin Microbiol Rev. 2016 Oct;29(4):915-26
pubmed: 27608937
Curr Comput Aided Drug Des. 2010 Mar;6(1):37-49
pubmed: 20370694
J Comput Chem. 2009 Dec;30(16):2785-91
pubmed: 19399780
Molecules. 2018 Feb 27;23(3):
pubmed: 29495447
J Proteome Res. 2015 Mar 6;14(3):1445-54
pubmed: 25664397
Mol Microbiol. 2007 Feb;63(4):1096-106
pubmed: 17238915
Nucleic Acids Res. 2009 Jan;37(Database issue):D499-508
pubmed: 18835847
BMC Bioinformatics. 2009 Jun 02;10:168
pubmed: 19486540
J Mol Graph Model. 2014 Feb;47:37-43
pubmed: 24316937
J Chem Inf Model. 2013 Sep 23;53(9):2409-22
pubmed: 23901876
Tuber Lung Dis. 1997;78(2):117-22
pubmed: 9692180
Nat Rev Drug Discov. 2011 Jun 24;10(7):507-19
pubmed: 21701501
Biochem Biophys Res Commun. 2017 Sep 30;491(4):1105-1111
pubmed: 28789944
Antimicrob Agents Chemother. 2009 Sep;53(9):3720-5
pubmed: 19528280
Drug Discov Today. 2006 Aug;11(15-16):741-8
pubmed: 16846802
Tuberculosis (Edinb). 2015 Mar;95(2):149-54
pubmed: 25547657
Microbiology (Reading). 2000 Feb;146 ( Pt 2):289-296
pubmed: 10708367
Curr Top Med Chem. 2010;10(1):127-41
pubmed: 19929824
J Med Chem. 2000 Dec 14;43(25):4759-67
pubmed: 11123984
Nucleic Acids Res. 2000 Jan 1;28(1):235-42
pubmed: 10592235
Mini Rev Med Chem. 2007 Feb;7(2):181-9
pubmed: 17305592
Chem Res Toxicol. 2021 May 17;34(5):1348-1354
pubmed: 33913699
J Comput Aided Mol Des. 2000 May;14(4):383-401
pubmed: 10815774
Biol Chem. 2011 Apr;392(4):277-89
pubmed: 21294681
Bioorg Chem. 2018 Oct;80:319-333
pubmed: 29986181
RSC Med Chem. 2020 Nov 6;11(12):1354-1365
pubmed: 34085044
Antimicrob Agents Chemother. 2015 Apr;59(4):2045-50
pubmed: 25605360
J Comput Chem. 2004 Sep;25(12):1463-73
pubmed: 15224390
Front Chem. 2020 Apr 28;8:343
pubmed: 32411671
J Biomol Struct Dyn. 2020 Jun;38(9):2521-2532
pubmed: 31244382
J Med Chem. 2007 Apr 19;50(8):1925-32
pubmed: 17367122
Nature. 2004 Dec 16;432(7019):862-5
pubmed: 15602552
Int J Mol Sci. 2019 Jun 06;20(11):
pubmed: 31174387
Molecules. 2020 May 27;25(11):
pubmed: 32471211
Proteins. 2003 Sep 1;52(4):609-23
pubmed: 12910460
Trends Biochem Sci. 1989 Jul;14(7):304-9
pubmed: 2672455
Bioinformatics. 2005 May 1;21(9):1908-16
pubmed: 15701681
J Biomol Struct Dyn. 2020 Jul;38(11):3396-3410
pubmed: 31422761
Drug Discov Today. 2016 Feb;21(2):288-98
pubmed: 26743596
J Chem Inf Model. 2012 Jul 23;52(7):1806-11
pubmed: 22758389
Molecules. 2020 Feb 04;25(3):
pubmed: 32033144
Antimicrob Agents Chemother. 2004 Aug;48(8):3006-9
pubmed: 15273113
Antimicrob Agents Chemother. 2009 May;53(5):2100-9
pubmed: 19237648
J Mol Biol. 1996 Aug 23;261(3):470-89
pubmed: 8780787
Trends Pharmacol Sci. 2008 Nov;29(11):576-81
pubmed: 18799223
J Biomol Struct Dyn. 2019 Mar;37(5):1254-1269
pubmed: 29557724
Trends Mol Med. 2011 Jan;17(1):25-33
pubmed: 21071272
J Chem Inf Model. 2012 Apr 23;52(4):867-81
pubmed: 22435959
Chembiochem. 2016 Dec 2;17(23):2264-2273
pubmed: 27653508
J Chem Inf Model. 2010 Feb 22;50(2):205-16
pubmed: 20088575
Int J Tuberc Lung Dis. 2003 Jan;7(1):6-21
pubmed: 12701830
Am J Ophthalmol. 2006 May;141(5):850-8
pubmed: 16546110
Mol Inform. 2021 May;40(5):e2000211
pubmed: 33283460
F1000Res. 2013 Sep 30;2:199
pubmed: 24555097
J Cheminform. 2017 May 4;9(1):27
pubmed: 29086046
Nat Rev Drug Discov. 2013 May;12(5):388-404
pubmed: 23629506
F1000Res. 2014 Mar 18;3:75
pubmed: 24741442
Org Biomol Chem. 2017 Dec 13;15(48):10245-10255
pubmed: 29182187
J Comput Aided Mol Des. 2012 Jan;26(1):13-4
pubmed: 22160556
PLoS One. 2017 Sep 5;12(9):e0183060
pubmed: 28873466
J Chem Inf Comput Sci. 2001 May-Jun;41(3):702-12
pubmed: 11410049
Nucleic Acids Res. 2010 Jul;38(Web Server issue):W582-9
pubmed: 20478829
Curr Med Chem. 2013;20(23):2839-60
pubmed: 23651302
Nat Med. 1996 Jun;2(6):662-7
pubmed: 8640557
Nucleic Acids Res. 2015 Jul 1;43(W1):W436-42
pubmed: 25956651
Nat Rev Drug Discov. 2005 Jan;4(1):45-58
pubmed: 15688072
Comb Chem High Throughput Screen. 2009 Dec;12(10):1000-16
pubmed: 20025565
J Comput Aided Mol Des. 1998 Jul;12(4):383-96
pubmed: 9777496
J Comput Chem. 2010 Jan 30;31(2):455-61
pubmed: 19499576
Appl Environ Microbiol. 2016 Jan 15;82(6):1958-1965
pubmed: 26773086
Clin Infect Dis. 2000 Feb;30(2):293-9
pubmed: 10671331
Antimicrob Agents Chemother. 2020 Aug 20;64(9):
pubmed: 32571810
Arch Pharm Res. 2017 Jun;40(6):676-694
pubmed: 28456911
BMC Infect Dis. 2015 Mar 25;15:153
pubmed: 25887373
Curr Protein Pept Sci. 2007 Aug;8(4):329-51
pubmed: 17696867
Bioorg Med Chem Lett. 2013 May 15;23(10):3096-100
pubmed: 23562055
J Enzyme Inhib Med Chem. 2016;31(sup2):201-207
pubmed: 27241561
J Antimicrob Chemother. 2011 Jul;66(7):1417-30
pubmed: 21558086
BMC Bioinformatics. 2010 Jul 12;11:374
pubmed: 20624289
J Mol Graph Model. 2015 Jul;60:124-31
pubmed: 26043661
Int J Mol Sci. 2019 Apr 26;20(9):
pubmed: 31027337
Ann Intern Med. 2016 Jul 19;165(2):125-33
pubmed: 27136449
J Antimicrob Chemother. 2011 Mar;66(3):564-73
pubmed: 21393229
J Antibiot (Tokyo). 2019 Oct;72(10):719-728
pubmed: 31292530
Curr Drug Metab. 2007 Dec;8(8):839-51
pubmed: 18220565
Curr Top Med Chem. 2014;14(16):1923-38
pubmed: 25262799
Sci Rep. 2017 Jul 5;7(1):4653
pubmed: 28680150
Arch Pharm (Weinheim). 2015 Mar;348(3):179-87
pubmed: 25690564
Bioorg Med Chem. 2016 Mar 1;24(5):1023-31
pubmed: 26822568
Methods Mol Biol. 2011;672:299-323
pubmed: 20838974
Tuberculosis (Edinb). 2012 Jan;92(1):72-83
pubmed: 21708485
Biochem Pharmacol. 2016 Apr 15;106:46-55
pubmed: 26867495
Drug Discov Today Technol. 2006 Autumn;3(3):307-13
pubmed: 24980533
Antibiotics (Basel). 2014 Jul 02;3(3):317-40
pubmed: 27025748
J Acquir Immune Defic Syndr. 2007 Oct 1;46(2):125-33
pubmed: 17721395
Bioorg Med Chem. 2016 Sep 15;24(18):4499-4508
pubmed: 27477207
AAPS J. 2012 Mar;14(1):133-41
pubmed: 22281989
Eur J Med Chem. 2018 Jul 15;155:754-763
pubmed: 29940465
Drug Discov Today. 2006 Feb;11(3-4):175-80
pubmed: 16533716
Future Microbiol. 2012 Jul;7(7):823-37
pubmed: 22827305
Curr Opin Pharmacol. 2018 Oct;42:81-94
pubmed: 30144650
Antimicrob Agents Chemother. 2008 Jun;52(6):2027-34
pubmed: 18378710
Int J Infect Dis. 2017 Mar;56:1-5
pubmed: 28232006
Drug Des Devel Ther. 2018 May 01;12:1065-1079
pubmed: 29750019
Antimicrob Agents Chemother. 2002 Sep;46(9):2765-71
pubmed: 12183226
Nucleic Acids Res. 2017 Jan 4;45(D1):D945-D954
pubmed: 27899562
J Chem Inf Model. 2011 Jun 27;51(6):1307-14
pubmed: 21604800
Eur J Med Chem. 2016 Oct 21;122:216-231
pubmed: 27371925
Science. 2004 Mar 19;303(5665):1813-8
pubmed: 15031495
Brief Bioinform. 2009 Sep;10(5):579-91
pubmed: 19433475
Mol Microbiol. 2008 Sep;69(5):1316-29
pubmed: 18651841
Sci Rep. 2016 Jun 10;6:27792
pubmed: 27283217
J Chem Inf Model. 2006 Mar-Apr;46(2):836-43
pubmed: 16563015
Proc Natl Acad Sci U S A. 2000 Aug 15;97(17):9677-82
pubmed: 10944230
Int J Infect Dis. 2021 Dec;113 Suppl 1:S96-S99
pubmed: 33713815
Microbiol Spectr. 2014 Aug;2(4):MGM2-0023-2013
pubmed: 26104205
ChemMedChem. 2008 Aug;3(8):1250-68
pubmed: 18663709
J Chem Inf Model. 2005 Sep-Oct;45(5):1369-75
pubmed: 16180913
mBio. 2017 Jan 17;8(1):
pubmed: 28096490
Eur J Pharmacol. 2009 Dec 25;625(1-3):90-100
pubmed: 19835861
J Med Chem. 2014 Jun 26;57(12):5293-305
pubmed: 24870926
Acta Trop. 2011 Jul;119(1):5-10
pubmed: 21515239
J Med Chem. 2004 May 6;47(10):2499-510
pubmed: 15115393
Antimicrob Agents Chemother. 2004 Feb;48(2):596-601
pubmed: 14742214
J Med Chem. 2015 Feb 26;58(4):2036-41
pubmed: 25658656
J Inorg Biochem. 2014 Mar;132:21-9
pubmed: 24188534
Nat Protoc. 2009;4(1):1-13
pubmed: 19131951
3 Biotech. 2021 Apr;11(4):204
pubmed: 33824847
Sci Rep. 2017 Mar 08;7:44116
pubmed: 28272524
J Chem Inf Model. 2015 Nov 23;55(11):2324-37
pubmed: 26479676
Curr Opin Chem Biol. 2017 Jun;38:117-126
pubmed: 28494316
Nucleic Acids Res. 2012 Apr;40(7):3018-30
pubmed: 22156370
J Chem Inf Model. 2011 Jun 27;51(6):1364-75
pubmed: 21618971
Nature. 2000 Jun 22;405(6789):962-6
pubmed: 10879539
Curr Top Med Chem. 2010;10(1):95-115
pubmed: 19929826
Biophys J. 2015 Jan 20;108(2):228-9
pubmed: 25606670
J Antibiot (Tokyo). 1953 Dec;6(4):182
pubmed: 13152032
J Mol Model. 2011 Jan;17(1):201-8
pubmed: 20383726
Drug Discov Today. 2011 Sep;16(17-18):831-9
pubmed: 21810482
J Antimicrob Chemother. 2009 Nov;64(5):1052-61
pubmed: 19734171
J Biomol Struct Dyn. 2011 Jun;28(6):907-17
pubmed: 21469751
Expert Opin Drug Discov. 2008 Aug;3(8):841-51
pubmed: 23484962
Protein Sci. 2018 Jan;27(1):129-134
pubmed: 28875543
Structure. 1996 Nov 15;4(11):1317-24
pubmed: 8939755
Antimicrob Agents Chemother. 2012 Apr;56(4):1797-809
pubmed: 22252828
J Med Chem. 2014 Jun 12;57(11):4487-97
pubmed: 24694071
Int J Appl Basic Med Res. 2013 Jan;3(1):1-2
pubmed: 23776831
Annu Rev Microbiol. 2007;61:35-50
pubmed: 18035606
Methods Mol Biol. 2011;716:23-38
pubmed: 21318898
Tuberculosis (Edinb). 2009 Sep;89(5):334-53
pubmed: 19758845
Antimicrob Agents Chemother. 2014;58(3):1479-87
pubmed: 24366731
Eur J Med Chem. 2015 Mar 6;92:401-14
pubmed: 25585006
Mol Microbiol. 2006 Dec;62(5):1220-7
pubmed: 17074073
J Antimicrob Chemother. 2003 Nov;52(5):790-5
pubmed: 14563891
Front Microbiol. 2013 Jul 23;4:208
pubmed: 23888158
J Natl Cancer Inst. 2011 Apr 6;103(7):553-61
pubmed: 21422402
Antimicrob Agents Chemother. 2005 Jun;49(6):2153-63
pubmed: 15917508
Arch Pharm Res. 2015 Sep;38(9):1686-701
pubmed: 26208641
Curr Pharm Des. 2016;22(5):572-81
pubmed: 26601966
Trends Microbiol. 2011 Feb;19(2):65-74
pubmed: 21129975
Pharmacol Rev. 2011 Mar;63(1):59-126
pubmed: 21228259
Nat Med. 2013 Sep;19(9):1157-60
pubmed: 23913123
Expert Opin Drug Discov. 2012 Oct;7(10):969-88
pubmed: 22860803
Microb Biotechnol. 2009 Jan;2(1):40-61
pubmed: 21261881
Molecules. 2017 Jan 17;22(1):
pubmed: 28106753
JAMA Intern Med. 2018 Nov 1;178(11):1451-1457
pubmed: 30264133
Cold Spring Harb Perspect Med. 2015 Apr 15;5(8):a021147
pubmed: 25877396
Nucleic Acids Res. 2012 Jul;40(Web Server issue):W387-92
pubmed: 22523085
Tuberculosis (Edinb). 2009 Mar;89(2):109-13
pubmed: 19249243