Discovery, X-ray structure and CPP-conjugation enabled uptake of p53/MDM2 macrocyclic peptide inhibitors.
Journal
RSC chemical biology
ISSN: 2633-0679
Titre abrégé: RSC Chem Biol
Pays: England
ID NLM: 101768727
Informations de publication
Date de publication:
02 Dec 2021
02 Dec 2021
Historique:
received:
16
03
2021
accepted:
21
08
2021
entrez:
3
1
2022
pubmed:
4
1
2022
medline:
4
1
2022
Statut:
epublish
Résumé
Mouse double minute 2 homolog (MDM2, Hdm2) is an important negative regulator of the tumor suppressor p53. Using a mRNA based display technique to screen a library of >10
Identifiants
pubmed: 34977581
doi: 10.1039/d1cb00056j
pii: d1cb00056j
pmc: PMC8637822
doi:
Types de publication
Journal Article
Langues
eng
Pagination
1661-1668Informations de copyright
This journal is © The Royal Society of Chemistry.
Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
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