Development of an mRNA replacement therapy for phenylketonuria.

LNP MT: Delivery Strategies PAH PKU hepatocytes lipid nanoparticle liver mRNA phenylketonuria replacement therapy

Journal

Molecular therapy. Nucleic acids
ISSN: 2162-2531
Titre abrégé: Mol Ther Nucleic Acids
Pays: United States
ID NLM: 101581621

Informations de publication

Date de publication:
14 Jun 2022
Historique:
received: 03 01 2022
accepted: 25 02 2022
entrez: 31 3 2022
pubmed: 1 4 2022
medline: 1 4 2022
Statut: epublish

Résumé

Phenylketonuria (PKU) is an inborn error caused by deficiencies in phenylalanine (Phe) metabolism. Mutations in the phenylalanine hydroxylase (PAH) gene are the main cause of the disease whose signature hallmarks of toxically elevated levels of Phe accumulation in plasma and organs such as the brain, result in irreversible intellectual disability. Here, we present a unique approach to treating PKU deficiency by using an mRNA replacement therapy. A full-length mRNA encoding human PAH (hPAH) is encapsulated in our proprietary lipid nanoparticle LUNAR and delivered to a

Identifiants

pubmed: 35356682
doi: 10.1016/j.omtn.2022.02.020
pii: S2162-2531(22)00048-8
pmc: PMC8933640
doi:

Types de publication

Journal Article

Langues

eng

Pagination

87-98

Informations de copyright

© 2022 The Authors.

Déclaration de conflit d'intérêts

The work included in this manuscript was performed using funds provided by Arcturus Therapeutics, Inc. The authors are current or former employees of Arcturus Therapeutics Inc.

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Auteurs

Carlos G Perez-Garcia (CG)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Ramon Diaz-Trelles (R)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Jerel Boyd Vega (JB)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Yanjie Bao (Y)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Marciano Sablad (M)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Patty Limphong (P)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Simon Chikamatsu (S)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Hailong Yu (H)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Wendy Taylor (W)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Priya P Karmali (PP)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Kiyoshi Tachikawa (K)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Padmanabh Chivukula (P)

Arcturus Therapeutics, Inc., 10628 Science Center Drive, Suite 250, San Diego, CA 92121, USA.

Classifications MeSH