Lithium salts as a treatment for COVID-19: Pre-clinical outcomes.


Journal

Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
ISSN: 1950-6007
Titre abrégé: Biomed Pharmacother
Pays: France
ID NLM: 8213295

Informations de publication

Date de publication:
May 2022
Historique:
received: 10 01 2022
revised: 20 03 2022
accepted: 23 03 2022
pubmed: 2 4 2022
medline: 28 4 2022
entrez: 1 4 2022
Statut: ppublish

Résumé

Identifying effective drugs for Coronavirus disease 2019 (COVID-19) is urgently needed. An efficient approach is to evaluate whether existing approved drugs have anti-SARS-CoV-2 effects. The antiviral properties of lithium salts have been studied for many years. Their anti-inflammatory and immune-potentiating effects result from the inhibition of glycogen synthase kinase-3. To obtain pre-clinical evidence on the safety and therapeutic effects of lithium salts in the treatment of COVID-19. Six different concentrations of lithium, ranging 2-12 mmol/L, were evaluated. Lithium inhibited the replication of SARS-CoV-2 virus in a dose-dependent manner with an IC These results provide pre-clinical evidence of the antiviral and immunotherapeutic effects of lithium against SARS-CoV-2, which supports an advance to clinical trials on COVID-19's patients.

Identifiants

pubmed: 35364381
pii: S0753-3322(22)00261-X
doi: 10.1016/j.biopha.2022.112872
pmc: PMC8947939
pii:
doi:

Substances chimiques

Antiviral Agents 0
Salts 0
Lithium 9FN79X2M3F

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

112872

Informations de copyright

Copyright © 2022 The Authors. Published by Elsevier Masson SAS.. All rights reserved.

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Auteurs

O Soriano-Torres (O)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba. Electronic address: ormany87@gmail.com.

E Noa Romero (E)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

N L González Sosa (NL)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

J M Enríquez Puertas (JM)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

A Fragas Quintero (A)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

M García Montero (M)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

D Martín Alfonso (D)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

Y Infante Hernández (Y)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

M Lastre (M)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

L Rodríguez-Pérez (L)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

Y Borrego (Y)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

V E González (VE)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

I G Vega (IG)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

R Ramos Pupo (R)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba; Biomedical Research Institute (BIOMED), Faculty of Medicine and Life Science, Hasselt University, Belgium.

L M Reyes (LM)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

M T Zumeta Dubé (MT)

Histology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

Amaro Hernández (A)

Histology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba.

I García de la Rosa (I)

Immunoassay Center, Havana, Cuba.

A Minguez Suárez (A)

MedSol Laboratories, Havana, Cuba.

L A Alarcón Camejo (LA)

MedSol Laboratories, Havana, Cuba.

M Rodríguez (M)

Civilian Defense Scientific Research Center, Mayabeque, Cuba.

R Oliva Hernández (R)

Finlay Vaccine Institute, Havana, Cuba.

C E Rudd (CE)

Centre de Recherche Maisonneuve-Rosemont Hospital (CR-HMR), Montreal, QC H1T 2M4, Canada; Département de Medicine, Université de Montréal, Montreal, QC H3C 3J7, Canada; Department of Medicine, Division of Endocrinology & Medical Biochemistry, McGill University Health Center, Canada.

O Pérez (O)

Immunology Department, Instituto de Ciencias Básicas y Preclínicas "Victoria de Girón", Universidad de Ciencias Médicas de La Habana, Havana, Cuba. Electronic address: oliver.perez@infomed.sld.cu.

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