Development of Bicyclo[3.1.0]hexane-Based A

Animals CHO Cells Cricetinae Hexanes Ligands Nucleosides / chemistry Radioligand Assay Receptor, Adenosine A3 / chemistry Structure-Activity Relationship
A3 receptors Adenosine receptors bicyclo[3.1.0]hexane methanocarba

Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
31 Mar 2022
Historique:
received: 09 03 2022
revised: 24 03 2022
accepted: 30 03 2022
entrez: 12 4 2022
pubmed: 13 4 2022
medline: 14 4 2022
Statut: epublish

Résumé

The adenosine A

Identifiants

DOI: 10.3390/molecules27072283 PMID: 35408685 PMC: PMC9000336
pubmed: 35408685
pii: molecules27072283
doi: 10.3390/molecules27072283
pmc: PMC9000336
pii:
doi:

Substances chimiques

Hexanes 0
Ligands 0
Nucleosides 0
Receptor, Adenosine A3 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Deutsche Forschungsgemeinschaft
ID : JU 2966/2-1
Organisme : National Institute of Health
ID : ZIADK-31117

Références

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pubmed: 15771421
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Auteurs

Jan Phillip Lemmerhirt (JP)

European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstr. 15, 48149 Münster, Germany.

Andreas Isaak (A)

European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstr. 15, 48149 Münster, Germany.

Rongfang Liu (R)

Leiden Academic Centre for Drug Research (LACDR), Division of Medicinal Chemistry, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.

Max Kock (M)

European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstr. 15, 48149 Münster, Germany.

Constantin G Daniliuc (CG)

Organisch-Chemisches Institut, University of Münster, Corrensstraße 40, 48149 Münster, Germany.
ORCID: 0000-0002-6709-3673

Kenneth A Jacobson (KA)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, MD 20892, USA.
ORCID: 0000-0001-8104-1493

Laura H Heitman (LH)

Leiden Academic Centre for Drug Research (LACDR), Division of Medicinal Chemistry, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
ORCID: 0000-0002-1381-8464

Anna Junker (A)

European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstr. 15, 48149 Münster, Germany.
ORCID: 0000-0001-5151-0930

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Classifications MeSH

questionsmedicales.fr › Eucaryotes › Animaux › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Cellules › Cellules épithéliales › Cellules CHO › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Rodentia › Muridae › Arvicolinae › Cricetinae › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Composés chimiques organiques › Hydrocarbures › Hydrocarbures acycliques › Alcanes › Hexanes › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Ligands › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Acides nucléiques, nucléotides et nucléosides › Nucléosides › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Techniques d'investigation › Techniques de laboratoire clinique › Dosage par compétition › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Protéines membranaires › Récepteurs de surface cellulaire › Récepteurs aux neuromédiateurs › Récepteurs purinergiques › Récepteurs purinergiques P1 › Récepteur A3 à l'adénosine › Development of Bicyclo[3.1.0]hexane-Based A
questionsmedicales.fr › Phénomènes physiologiques › Phénomènes pharmacologiques et toxicologiques › Phénomènes pharmacologiques › Relation structure-activité › Development of Bicyclo[3.1.0]hexane-Based A