Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437.


Journal

ACS chemical biology
ISSN: 1554-8937
Titre abrégé: ACS Chem Biol
Pays: United States
ID NLM: 101282906

Informations de publication

Date de publication:
20 05 2022
Historique:
pubmed: 29 4 2022
medline: 24 5 2022
entrez: 28 4 2022
Statut: ppublish

Résumé

Anandamide or

Identifiants

pubmed: 35482948
doi: 10.1021/acschembio.2c00122
pmc: PMC9127799
doi:

Substances chimiques

Arachidonic Acids 0
Endocannabinoids 0
Polyunsaturated Alkamides 0
anandamide UR5G69TJKH

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1174-1183

Références

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Auteurs

Berend Gagestein (B)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Anna F Stevens (AF)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Domenico Fazio (D)

European Center for Brain Research/IRCCS Santa Lucia Foundation, Via del Fosso di Fiorano 64, Rome 00143, Italy.

Bogdan I Florea (BI)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Tom van der Wel (T)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Alexander T Bakker (AT)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Filomena Fezza (F)

Department of Experimental Medicine, Tor Vergata University of Rome, Via Montpellier 1, Rome 00121, Italy.

Hans den Dulk (HD)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Herman S Overkleeft (HS)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

Mauro Maccarrone (M)

European Center for Brain Research/IRCCS Santa Lucia Foundation, Via del Fosso di Fiorano 64, Rome 00143, Italy.
Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, Via Vetoio snc, 67100 L'Aquila, Italy.

Mario van der Stelt (M)

Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University, Einsteinweg 55, Leiden 2333 CC, The Netherlands.

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Classifications MeSH