Mosquitocidal efficacy of embelin and its derivatives against Aedes aegypti L. and Culex quinquefasciatus Say. (Diptera: Culicidae) and computational analysis of acetylcholinesterase 1 (AChE1) inhibition.

Acetylcholinesterase Aedes Animals Benzoquinones Culex Larva Molecular Docking Simulation Plant Extracts / pharmacology
Aedes aegypti Culex quinquefasciatus Derivatives Embelin Molecular docking Molecular dynamics Mosquitocidal efficacy

Journal

Computers in biology and medicine
ISSN: 1879-0534
Titre abrégé: Comput Biol Med
Pays: United States
ID NLM: 1250250

Informations de publication

Date de publication:
07 2022
Historique:
received: 10 03 2022
revised: 13 04 2022
accepted: 14 04 2022
pubmed: 30 4 2022
medline: 25 6 2022
entrez: 29 4 2022
Statut: ppublish

Résumé

Embelin was isolated from the chloroform extract of Embelia ribes (Burm.f.) fruits; its derivative compounds 6-bromoembelin and vilangin were prepared, and they were evaluated for mosquitocidal activities against the third instar larvae and pupae of Aedes aegypti L. and Culex quinquefasciatus Say. (Diptera: Culicidae). The concentrations used were 0.5, 1.0, 1.5, and 2.0 ppm. Embelin recorded LC

Identifiants

DOI: 10.1016/j.compbiomed.2022.105535 PMID: 35487124
pubmed: 35487124
pii: S0010-4825(22)00327-4
doi: 10.1016/j.compbiomed.2022.105535
pii:
doi:

Substances chimiques

Benzoquinones 0
Plant Extracts 0
Acetylcholinesterase EC 3.1.1.7
embelin SHC6U8F5ER

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

105535

Informations de copyright

Copyright © 2022 Elsevier Ltd. All rights reserved.

Auteurs

Antony Stalin (A)

Institute of Fundamental and Frontier Sciences, University of Electronic Science and Technology of China, Chengdu, 610 054, China. Electronic address: a.staanlin@gmail.com.

Appadurai Daniel Reegan (A)

National Centre for Disease Control, Bengaluru Branch, No:8, NTI Campus, Bellary Road, Bengaluru, 560 003, Karnataka, India; Xavier Research Foundation, St. Xavier's College, Affiliated to the Manonmaniam Sundaranar University, Palayamkottai, 627 002, Tamil Nadu, India. Electronic address: danielreegan85@gmail.com.

Munusamy Rajiv Gandhi (M)

National Biodiversity Authority, 5th Floor, CSIR Road, TICEL Bio Park, Taramani, Chennai, 600 113, India.

R R Saravanan (RR)

Department of Physics, Meenakshi Chandrasekaran College of Arts and Science, Karambayam, Pattukkottai, Thanjavur, 614 626, India.

Kedike Balakrishna (K)

Entomology Research Institute, Loyola College, Affiliated to the University of Madras, Chennai, 600 034, Tamil Nadu, India.

Abd El-Latif Hesham (AE)

Genetics Department, Faculty of Agriculture, Beni-Suef University, Beni-Suef, 62511, Egypt.

Savarimuthu Ignacimuthu (S)

Xavier Research Foundation, St. Xavier's College, Affiliated to the Manonmaniam Sundaranar University, Palayamkottai, 627 002, Tamil Nadu, India.

Ying Zhang (Y)

Department of Anesthesiology, Hospital (T.C.M) Affiliated To Southwest Medical University, Luzhou, China. Electronic address: zhangying021210@163.com.

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Classifications MeSH

questionsmedicales.fr › Enzymes et coenzymes › Enzymes › Hydrolases › Esterases › Carboxylic ester hydrolases › Cholinesterases › Acetylcholinesterase › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Eucaryotes › Animaux › Invertébrés › Arthropodes › Insectes › Pterygota › Neoptera › Holometabola › Diptera › Nematocera › Culicomorpha › Culicidae › Aedes › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Eucaryotes › Animaux › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Composés chimiques organiques › Quinones › Benzoquinones › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Eucaryotes › Animaux › Invertébrés › Arthropodes › Insectes › Pterygota › Neoptera › Holometabola › Diptera › Nematocera › Culicomorpha › Culicidae › Culex › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Phénomènes physiologiques › Croissance et développement › Morphogenèse › Métamorphose biologique › Étapes du cycle de vie › Larve › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Sciences de l'information › Méthodologies informatiques › Simulation numérique › Simulation de docking moléculaire › Mosquitocidal efficacy of embelin and its...
questionsmedicales.fr › Préparations pharmaceutiques › Extraits de plantes › Mosquitocidal efficacy of embelin and its...