The role of progesterone receptor membrane component (PGRMC) in the endometrium.


Journal

Steroids
ISSN: 1878-5867
Titre abrégé: Steroids
Pays: United States
ID NLM: 0404536

Informations de publication

Date de publication:
08 2022
Historique:
received: 28 03 2022
revised: 25 04 2022
accepted: 02 05 2022
pubmed: 9 5 2022
medline: 29 6 2022
entrez: 8 5 2022
Statut: ppublish

Résumé

PGRMC is a non-classical receptor that mediates the non-genomic responses to progesterone and is distributed in different subcellular compartments. PGRMC belongs to the membrane-associated progesterone receptor (MAPR) family. Two PGRMC subtypes (PGRMC1 and PGRMC2) have been characterized, and both are expressed in the human endometrium. PGRMC expression is differentially regulated during the menstrual cycle in the human endometrium. Although PGRMC1 is predominantly expressed in the proliferative phase and PGRMC2 in the secretory phase, this expression changes in pathologies such as endometriosis, in which PGRMC2 expression considerably decreases, promoting progesterone resistance. In endometrial cancer, PGRMC1 is overexpressed, its activation induces tumors growth, and confers chemoresistance in the presence of progesterone. Thus, PGRMCs play a key role in progesterone actions in the endometrium.

Identifiants

pubmed: 35526781
pii: S0039-128X(22)00078-2
doi: 10.1016/j.steroids.2022.109040
pii:
doi:

Substances chimiques

Membrane Proteins 0
PGRMC1 protein, human 0
PGRMC2 protein, human 0
Receptors, Progesterone 0
Progesterone 4G7DS2Q64Y

Types de publication

Journal Article Review Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

109040

Informations de copyright

Copyright © 2022 Elsevier Inc. All rights reserved.

Auteurs

Dora Maria Velázquez Hernández (DM)

Unidad de Investigación en Reproducción Humana, Instituto Nacional de Perinatología-Facultad de Química, Universidad Nacional Autónoma de México, Mexico City, Mexico.

Edgar Ricardo Vázquez-Martínez (ER)

Unidad de Investigación en Reproducción Humana, Instituto Nacional de Perinatología-Facultad de Química, Universidad Nacional Autónoma de México, Mexico City, Mexico.

Ignacio Camacho-Arroyo (I)

Unidad de Investigación en Reproducción Humana, Instituto Nacional de Perinatología-Facultad de Química, Universidad Nacional Autónoma de México, Mexico City, Mexico. Electronic address: camachoarroyo@gmail.com.

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Classifications MeSH