A strained alkyne-containing bipyridine reagent; synthesis, reactivity and fluorescence properties.


Journal

RSC advances
ISSN: 2046-2069
Titre abrégé: RSC Adv
Pays: England
ID NLM: 101581657

Informations de publication

Date de publication:
04 Nov 2019
Historique:
received: 29 08 2019
accepted: 29 10 2019
entrez: 11 5 2022
pubmed: 6 11 2019
medline: 6 11 2019
Statut: epublish

Résumé

We report the synthesis of a bipyridyl reagent containing a strained alkyne, which significantly restricts its flexibility. Upon strain-promoted alkyne-azide cycloaddition (SPAAC) with an azide, which does not require a Cu catalyst, the structure becomes significantly more flexible and an increase in fluorescence is observed. Upon addition of Zn(ii), the fluorescence is enhanced further. The reagent has the potential to act as a fluorescent labelling agent with azide-containing substrates, including biological molecules.

Identifiants

pubmed: 35540623
doi: 10.1039/c9ra06866j
pii: c9ra06866j
pmc: PMC9074932
doi:

Types de publication

Journal Article

Langues

eng

Pagination

36154-36161

Informations de copyright

This journal is © The Royal Society of Chemistry.

Déclaration de conflit d'intérêts

The authors declare no conflicting interests.

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Auteurs

Sam Forshaw (S)

Department of Chemistry, The University of Warwick Coventry CV4 7AL UK m.wills@warwick.ac.uk.

Richard C Knighton (RC)

Department of Chemistry, The University of Warwick Coventry CV4 7AL UK m.wills@warwick.ac.uk.

Jami Reber (J)

Department of Chemistry, The University of Warwick Coventry CV4 7AL UK m.wills@warwick.ac.uk.

Jeremy S Parker (JS)

Early Chemical Development, Pharmaceutical Sciences, IMED Biotech Unit, AstraZeneca Macclesfield SK10 2NA UK.

Nikola P Chmel (NP)

Department of Chemistry, The University of Warwick Coventry CV4 7AL UK m.wills@warwick.ac.uk.

Martin Wills (M)

Department of Chemistry, The University of Warwick Coventry CV4 7AL UK m.wills@warwick.ac.uk.

Classifications MeSH