From Antarctica to cancer research: a novel human DNA topoisomerase 1B inhibitor from Antarctic sponge
Natural product
cancer
drug development
topoisomerase
Journal
Journal of enzyme inhibition and medicinal chemistry
ISSN: 1475-6374
Titre abrégé: J Enzyme Inhib Med Chem
Pays: England
ID NLM: 101150203
Informations de publication
Date de publication:
Dec 2022
Dec 2022
Historique:
entrez:
23
5
2022
pubmed:
24
5
2022
medline:
25
5
2022
Statut:
ppublish
Résumé
Nature has been always a great source of possible lead compounds to develop new drugs against several diseases. Here we report the identification of a natural compound, membranoid G, derived from the Antarctic sponge
Identifiants
pubmed: 35603503
doi: 10.1080/14756366.2022.2078320
pmc: PMC9132426
doi:
Substances chimiques
Antineoplastic Agents
0
Topoisomerase Inhibitors
0
DNA
9007-49-2
DNA Topoisomerases, Type I
EC 5.99.1.2
DNA Topoisomerases, Type II
EC 5.99.1.3
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
1404-1410Références
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