Linear and branched polymer prodrugs of the water-soluble nucleoside reverse-transcriptase inhibitor emtricitabine as structural materials for long-acting implants.


Journal

Journal of materials chemistry. B
ISSN: 2050-7518
Titre abrégé: J Mater Chem B
Pays: England
ID NLM: 101598493

Informations de publication

Date de publication:
15 06 2022
Historique:
pubmed: 24 5 2022
medline: 18 6 2022
entrez: 23 5 2022
Statut: epublish

Résumé

Long-acting drug delivery is a growing area of interest as it overcomes many challenges related to patient adherence to therapy and the pill burden associated with chronic illness. Injectable formulations are becoming more common and drug-releasing implants also provide several opportunities. Highly water soluble drug compounds are poor candidates for long-acting delivery. Here, the water-soluble nucleoside reverse transcriptase inhibitor emtricitabine (FTC) has been used as a novel A-B monomer in step-growth polymerisation with chloroformate functional C

Identifiants

pubmed: 35604111
doi: 10.1039/d2tb00825d
pmc: PMC9199480
doi:

Substances chimiques

Anti-HIV Agents 0
Nucleosides 0
Polymers 0
Prodrugs 0
Reverse Transcriptase Inhibitors 0
Water 059QF0KO0R
DNA-Directed RNA Polymerases EC 2.7.7.6
Emtricitabine G70B4ETF4S

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

4395-4404

Subventions

Organisme : NIAID NIH HHS
ID : R01 AI134091
Pays : United States

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Auteurs

Anika Shakil (A)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

Faye Y Hern (FY)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

Chung Liu (C)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

Kartik Temburnikar (K)

Department of Pharmacology and Molecular Sciences, The Johns Hopkins University School of Medicine, 725 North Wolfe St., Baltimore, MD, 21205, USA.

Pierre Chambon (P)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

Neill Liptrott (N)

Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.
Department of Pharmacology and Therapeutics, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool, L7 3NY, UK.

Tom O McDonald (TO)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

Megan Neary (M)

Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.
Department of Pharmacology and Therapeutics, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool, L7 3NY, UK.

Andrew Owen (A)

Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.
Department of Pharmacology and Therapeutics, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool, L7 3NY, UK.

Caren Freel Meyers (C)

Department of Pharmacology and Molecular Sciences, The Johns Hopkins University School of Medicine, 725 North Wolfe St., Baltimore, MD, 21205, USA.

Steve P Rannard (SP)

Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, UK. srannard@liverpool.ac.uk.
Materials Innovation Factory, University of Liverpool, Crown Street, L69 7ZD, UK.
Centre of Excellence in Long-acting Therapeutics (CELT), University of Liverpool, Liverpool, L7 3NY, UK.

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