Optimization of the Synthesis of Natural Polymeric Nanoparticles of Inulin Loaded with Quercetin: Characterization and Cytotoxicity Effect.

flavonoid inulin nanoparticle quercetin

Journal

Pharmaceutics
ISSN: 1999-4923
Titre abrégé: Pharmaceutics
Pays: Switzerland
ID NLM: 101534003

Informations de publication

Date de publication:
19 Apr 2022
Historique:
received: 10 03 2022
revised: 04 04 2022
accepted: 07 04 2022
entrez: 28 5 2022
pubmed: 29 5 2022
medline: 29 5 2022
Statut: epublish

Résumé

Quercetin is a bioactive component that is capable of having therapeutic potential in the prevention of different noncommunicable chronic diseases (NCDs). However, it presents instability in the gastrointestinal tract in addition to low bioavailability. One way to overcome the limitations of quercetin lies in using nanotechnology for the development of nanoparticles, based on biopolymers, that are capable of being ingestible. Inulin, a fructan-type polysaccharide, acts as a delivery system for the release of quercetin in a target cell, guaranteeing the stability of the molecule. Inulin-coated quercetin nanoparticles were synthesized by the spray dryer method, and four variables were evaluated, namely inulin concentration (5-10%

Identifiants

pubmed: 35631474
pii: pharmaceutics14050888
doi: 10.3390/pharmaceutics14050888
pmc: PMC9147723
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Monterrey Institute of Technology and Higher Education
ID : APC

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Auteurs

Jocelyn C Ayala-Fuentes (JC)

Tecnológico de Monterrey, Escuela de Ingeniería y Ciencias, Ave. Eugenio Garza Sada 2501 Sur, Monterrey 64849, Mexico.

Melissa Zulahi Gallegos-Granados (MZ)

Facultad de Ciencias Químicas e Ingeniería, Universidad Autónoma de Baja California, Tijuana 22260, Mexico.

Luis Jesús Villarreal-Gómez (LJ)

Facultad de Ciencias Químicas e Ingeniería, Universidad Autónoma de Baja California, Tijuana 22260, Mexico.
Facultad de Ciencias de la Ingeniería y Tecnología, Universidad Autónoma de Baja California, Tijuana 22260, Mexico.

Marilena Antunes-Ricardo (M)

Tecnologico de Monterrey, The Institute for Obesity Research, Ave. Eugenio Garza Sada 2501 Sur, Monterrey 64849, Mexico.

Daniel Grande (D)

Univ Est Creteil, CNRS, Institut de Chimie et des Matériaux Paris-Est (ICMPE), 2, rue Henri Du-nant, 94320 Thiais, France.

Rocio Alejandra Chavez-Santoscoy (RA)

Tecnológico de Monterrey, Escuela de Ingeniería y Ciencias, Ave. Eugenio Garza Sada 2501 Sur, Monterrey 64849, Mexico.

Classifications MeSH