A Two Amino Acid Duplication, L167E168, in the Ω-Loop Drastically Decreases Carbapenemase Activity of KPC-53, a Natural Class A β-Lactamase.


Journal

Antimicrobial agents and chemotherapy
ISSN: 1098-6596
Titre abrégé: Antimicrob Agents Chemother
Pays: United States
ID NLM: 0315061

Informations de publication

Date de publication:
21 06 2022
Historique:
pubmed: 2 6 2022
medline: 24 6 2022
entrez: 1 6 2022
Statut: ppublish

Résumé

KPC-53 enzyme is a natural KPC variant which showed a duplication of L167E168 residues in the Ω-loop structure. The

Identifiants

pubmed: 35647648
doi: 10.1128/aac.02402-21
pmc: PMC9211410
doi:

Substances chimiques

Amino Acids 0
Anti-Bacterial Agents 0
Azabicyclo Compounds 0
Bacterial Proteins 0
Drug Combinations 0
beta-Lactamase Inhibitors 0
beta-Lactamases EC 3.5.2.6
carbapenemase EC 3.5.2.6

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

e0240221

Références

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Auteurs

Alessandra Piccirilli (A)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Sabrina Cherubini (S)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Giuseppe Celenza (G)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Gian Maria Rossolini (GM)

Department of Experimental and Clinical Medicine, University of Florence, Florence, Italy.
Clinical Microbiology and Virology Unit, Florence Careggi University Hospital, Florence Italy.

Fabrizia Brisdelli (F)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Bernardetta Segatore (B)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Luigi Principe (L)

Clinical Microbiology and Virology Unit, A. Manzoni Hospital, Lecco, Italy.

Francesco Luzzaro (F)

Clinical Microbiology and Virology Unit, A. Manzoni Hospital, Lecco, Italy.

Lilia Andriani (L)

Clinical Pathology and Microbiology Unit, Moriggia Pelascini General Hospital, Gravedona, Italy.

Gianfranco Amicosante (G)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

Mariagrazia Perilli (M)

Department of Biotechnological and Applied Clinical Sciences, University of L'Aquila, L'Aquila, Italy.

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Classifications MeSH